Target Details
| UniProt AC | Q9UEE5 |
|---|---|
| Gene Symbol | STK17A |
| Protein Name | Serine/threonine-protein kinase 17A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 277
- Clinical molecules 13
- Avg pChEMBL 6.99
Active Molecules (277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WINHZLLDWRZWRT
|
9.0 | Kd | 201 | Yes | |
HKSZLNNOFSGOKW
|
8.6 | Ki | 118 | — | |
YYLKKYCXAOBSRM
|
8.5 | Kd | 191 | — | |
RYYNGWLOYLRZLK
|
8.5 | Ki | 104 | — | |
ZKLJKKASNXVQBZ
|
8.5 | Ki | 27 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
GCYXEGSPUDSZJY
|
8.4 | Ki | 82 | — | |
ZSZOBRBJIJWWHH
|
8.3 | IC50 | 4 | — | |
WEFRCKPVMWDRAK
|
8.3 | Kd | 5 | — | |
KHGPYYFCIAISBU
|
8.2 | Ki | 31 | — | |
DPEXRCOBPACFOO
|
8.1 | Ki | 36 | — | |
RWKDVIAVTRRJIR
|
8.1 | Ki | 23 | — | |
XNWKXXIGSPPPBH
|
8.1 | Ki | 31 | — | |
UOPCRSIUYMGQCP
|
8.1 | Kd | 6 | — | |
CNCRCDLWUGCPSJ
|
8.0 | IC50 | 5 | — | |
LOLPPWBBNUVNQZ
|
8.0 | IC50 | 97 | Yes | |
SYMILEXMAHCATG
|
8.0 | Kd | 4 | — | |
UDFDIIVNIYWXDM
|
8.0 | Ki | 74 | — | |
SOJKVKSSTDCNFB
|
8.0 | IC50 | 2 | — | |
IDNFFZUHFOQNRQ
|
7.9 | IC50 | 2 | — | |
XKQNBVAZAFAZFL
|
7.9 | IC50 | 6 | — | |
FQEODTMNWMDUMD
|
7.9 | Ki | 25 | — | |
UYGYYOIUVFMGKQ
|
7.9 | Ki | 30 | — | |
WYOMXSAYYXBPMN
|
7.9 | Ki | 24 | — | |
XZONYYFHQICDAM
|
7.9 | Ki | 19 | — | |
HHLFERIUOTYKKU
|
7.9 | Kd | 2 | — | |
GOYAADNAKVCRJS
|
7.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
PFZRXJIYAFANHP
|
7.8 | IC50 | 4 | — | |
CCQLYJZEWHWASR
|
7.8 | IC50 | 5 | — | |
DPMDOFDIFNBKGS
|
7.8 | IC50 | 2 | — | |
BEJCLDKQCNVTQR
|
7.8 | Ki | 16 | — | |
BSFNGHCTZDCQBF
|
7.8 | Ki | 93 | — | |
IODFDZLIZNZVAP
|
7.8 | IC50 | 2 | — | |
IZAVTOABECKIDH
|
7.8 | Ki | 20 | — | |
RFBPWKMQWSIPEO
|
7.8 | Ki | 28 | — | |
XXSPHNFKLDJDAK
|
7.8 | Ki | 26 | — | |
YZVSEVMXAIJHKO
|
7.8 | IC50 | 2 | — | |
VCZRYZZCLOMGOV
|
7.8 | IC50 | 4 | — | |
GTVLFJMUKIZPEJ
|
7.7 | IC50 | 2 | — | |
KAEJBHCXBMUJRI
|
7.7 | IC50 | 2 | — | |
UOUMREPCEXJVFD
|
7.7 | IC50 | 2 | — | |
NLUPJKQOKWBWFC
|
7.7 | Ki | 69 | — | |
RFVBRKXQYUDGIO
|
7.7 | Ki | 23 | — | |
VUQUBDXLGAPBGS
|
7.7 | IC50 | 2 | — | |
WZISGNDZZPSYRP
|
7.7 | Ki | 20 | — | |
XOCCIJUVHIYNCB
|
7.7 | IC50 | 2 | — | |
AHQYMFOEOWUTJB
|
7.7 | IC50 | 2 | — | |
GGNAPCQTOZTGTK
|
7.7 | IC50 | 2 | — | |
YQMFNWQNASFQAE
|
7.7 | IC50 | 5 | — |