Target Details
| UniProt AC | Q9UBY5 |
|---|---|
| Gene Symbol | LPAR3 |
| Protein Name | Lysophosphatidic acid receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 36
- Clinical molecules 0
- Avg pChEMBL 6.81
KEGG Pathways (5)
Active Molecules (36)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUXSKJSPPDINEH
|
8.1 | IC50 | 3 | — | |
AEFXZQBYWHGBOY
|
7.5 | IC50 | 2 | — | |
WFNXESYFHAMZSY
|
7.4 | IC50 | 2 | — | |
HVANCKKENVXQOH
|
7.4 | Ki | 2 | — | |
IXNPTKKSRPZDOX
|
7.4 | Ki | 2 | — | |
QGFGIQUXZJXHPN
|
7.4 | IC50 | 2 | — | |
FFMZNYWFUDQTJJ
|
7.3 | Ki | 2 | — | |
SPTAXSFFLMLIAF
|
7.3 | Ki | 2 | — | |
LKYKLVDCGBTNJZ
|
7.3 | IC50 | 2 | — | |
XYSBQYUENLDGMI
|
7.2 | IC50 | 2 | — | |
VKPRWVOYFUXFAT
|
7.2 | IC50 | 2 | — | |
IKJZZCLSUSZHFO
|
7.2 | IC50 | 2 | — | |
GDLXQEKNJMCXRS
|
7.1 | IC50 | 2 | — | |
HKSCEHNRNXWQAZ
|
6.9 | IC50 | 2 | — | |
XYSBQYUENLDGMI
|
6.8 | IC50 | 2 | — | |
HLVKVWDSLLFMSX
|
6.8 | Ki | 4 | — | |
JGCATLCTRCCGRP
|
6.8 | Ki | 4 | — | |
XHZMTTZICDAOHN
|
6.8 | IC50 | 2 | — | |
PLCCQSPJUXGEHV
|
6.7 | IC50 | 2 | — | |
LLIFMNUXGDHTRO
|
6.7 | IC50 | 2 | — | |
XXIOBZYOOQRDDS
|
6.7 | IC50 | 2 | — | |
VNBIUEOBRLCNQI
|
6.6 | IC50 | 2 | — | |
HKSCEHNRNXWQAZ
|
6.5 | IC50 | 2 | — | |
HZFPOTBCYPWQSH
|
6.5 | Ki | 2 | — | |
KYUUSQMQCHIHII
|
6.5 | IC50 | 2 | — | |
VTJPSPQBNJNSKO
|
6.5 | IC50 | 2 | — | |
HFYPTENHTPNXGP
|
6.4 | IC50 | 3 | — | |
CSFMYMIHKKPMPF
|
6.4 | Ki | 2 | — | |
WKODFGZRSIFURU
|
6.3 | IC50 | 2 | — | |
ZNPWHDPODRSYQC
|
6.3 | IC50 | 2 | — | |
PHXJFMYKLBONBN
|
6.3 | Ki | 2 | — | |
YGXPAGSHLFJKFV
|
6.2 | Ki | 2 | — | |
YZILIQNNTIKUCA
|
6.2 | Ki | 2 | — | |
WFNXESYFHAMZSY
|
6.2 | IC50 | 2 | — | |
SWATWOUWJLKSFA
|
6.1 | IC50 | 2 | — | |
XHZMTTZICDAOHN
|
6.0 | IC50 | 2 | — |