Target Details
| UniProt AC | Q9UBS5 |
|---|---|
| Gene Symbol | GABBR1 |
| Protein Name | Gamma-aminobutyric acid type B receptor subunit 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF00084 (Sushi) |
Summary
- Multi-target molecules 27
- Clinical molecules 0
- Avg pChEMBL 7.49
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FDGOGCVLTKRRTJ
|
9.7 | IC50 | 2 | — | |
PJKJUMXCCOXVCF
|
8.9 | IC50 | 2 | — | |
FIQKPIGOFVCVTG
|
8.6 | IC50 | 4 | — | |
ZTHNRNOOZGJLRR
|
8.6 | IC50 | 2 | — | |
JGGVBBYJRQOPPA
|
8.4 | IC50 | 2 | — | |
CPIMXZAMIJJWLD
|
8.3 | IC50 | 4 | — | |
NHVRIDDXGZPJTJ
|
8.2 | IC50 | 3 | — | |
VSRMCPVTOJHMJM
|
7.9 | IC50 | 2 | — | |
KPYSYYIEGFHWSV
|
7.8 | IC50 | 2 | — | |
UROJZRVINWISIJ
|
7.8 | IC50 | 2 | — | |
CFTHWIIIZOVWJE
|
7.7 | IC50 | 2 | — | |
JXPXSJRYIIVYSJ
|
7.7 | IC50 | 2 | — | |
QLIIRQZTJJMJDY
|
7.7 | IC50 | 2 | — | |
RJOBXTDLIMOTCT
|
7.6 | IC50 | 2 | — | |
BTCSSZJGUNDROE
|
7.6 | IC50 | 23 | — | |
FUUPFUIGNBPCAY
|
7.5 | IC50 | 2 | — | |
KPYSYYIEGFHWSV
|
7.5 | IC50 | 2 | — | |
RWZSGLLMGBEMNE
|
7.4 | IC50 | 2 | — | |
CCFBFTKQKRGULP
|
6.8 | IC50 | 2 | — | |
NRAKQMOQGMIXRK
|
6.7 | IC50 | 2 | — | |
YOPOCOPYSKJKCU
|
6.5 | IC50 | 2 | — | |
NAMMMMPTLWTBHY
|
6.4 | IC50 | 2 | — | |
KMZGFUXQKZETKC
|
6.3 | IC50 | 2 | — | |
CDFQDLUHBLZCGL
|
6.2 | IC50 | 2 | — | |
XYDCKPSWUYIZGR
|
6.1 | IC50 | 2 | — | |
UQSUKRWHUNWKRZ
|
6.1 | IC50 | 2 | — | |
RZRFDYWPDLJLMD
|
6.0 | IC50 | 2 | — |