Target Details
| UniProt AC | Q9UBL3 |
|---|---|
| Gene Symbol | ASH2L |
| Protein Name | Set1/Ash2 histone methyltransferase complex subunit ASH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21198 (ASH2L-like_WH) PF21257 (PHD_ash2p_like) PF00622 (SPRY) |
Summary
- Multi-target molecules 35
- Clinical molecules 0
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NNIBWLKDWXOMEW
|
7.9 | IC50 | 5 | — | |
ZAIPJVQTYUSDTG
|
7.9 | IC50 | 5 | — | |
ZNCYDGWICNBNGY
|
7.8 | IC50 | 5 | — | |
BAWZTNUTCPWRFJ
|
7.7 | IC50 | 5 | — | |
HWBBSTOZNJTCST
|
7.6 | IC50 | 5 | — | |
WNZPPUDGOCDFHQ
|
7.5 | IC50 | 5 | — | |
RSWJWQUYPRQBFS
|
7.3 | IC50 | 5 | — | |
BNFSVXBSRYHZTB
|
7.2 | IC50 | 5 | — | |
AAAQFGUYHFJNHI
|
7.2 | IC50 | 252 | — | |
KJOQVBZBXKPYJX
|
7.2 | IC50 | 5 | — | |
NPFRAPJTDVLBBW
|
7.1 | IC50 | 5 | — | |
PRAJCBYVBKZLED
|
7.1 | IC50 | 5 | — | |
XCVJSTZYHUNTCU
|
7.0 | IC50 | 5 | — | |
AMSVGXDFPHGXFJ
|
6.9 | IC50 | 5 | — | |
KXYGAIVJVQJFDQ
|
6.9 | IC50 | 5 | — | |
MWWRLWPCGQFTIQ
|
6.9 | IC50 | 5 | — | |
OXSOFPMSKVUQBE
|
6.9 | IC50 | 5 | — | |
JGIIYJOEBDGPQO
|
6.9 | IC50 | 5 | — | |
VHPRRJZGFMSHQV
|
6.9 | IC50 | 5 | — | |
UWACKSCSSLOEGH
|
6.8 | IC50 | 5 | — | |
JBLHDYOCJVQGEP
|
6.7 | IC50 | 5 | — | |
PVXYYWORFYROCX
|
6.7 | IC50 | 4 | — | |
QTSKXZZDLJLJLM
|
6.7 | IC50 | 5 | — | |
DHBHJVJPRVYFCA
|
6.7 | IC50 | 5 | — | |
RNNUHFXCYYPDIF
|
6.6 | IC50 | 5 | — | |
CZWZZEUKNASAHM
|
6.5 | IC50 | 4 | — | |
SILRGLDFBXVGOQ
|
6.5 | IC50 | 5 | — | |
JZOSRTPOYRYTRA
|
6.3 | IC50 | 5 | — | |
SUXNCBRCYTZFPW
|
6.3 | IC50 | 5 | — | |
ZAIPJVQTYUSDTG
|
6.3 | IC50 | 5 | — | |
RZKSQRIPRKWVBU
|
6.3 | IC50 | 4 | — | |
BCIPILGGOSCOMC
|
6.2 | IC50 | 5 | — | |
RPXXFSOUEYJZLT
|
6.2 | IC50 | 5 | — | |
ZJUKTBDSGOFHSH
|
6.1 | IC50 | 22 | — | |
CMZXXROIVBWQKJ
|
6.1 | IC50 | 5 | — |