Target Details
| UniProt AC | Q9UBF8 |
|---|---|
| Gene Symbol | PI4KB |
| Protein Name | Phosphatidylinositol 4-kinase beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF21245 (PI4KB-PIK1_PIK) |
Summary
- Multi-target molecules 90
- Clinical molecules 14
- Avg pChEMBL 6.52
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (90)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTQOHJNXDAUMOA
|
6.3 | IC50 | 13 | Yes | |
QATDLTPQGNUUQD
|
6.2 | IC50 | 4 | — | |
GLWWXTJSWUKLBH
|
6.2 | IC50 | 4 | — | |
LEWJWUJNURRNQY
|
6.2 | IC50 | 4 | — | |
PPECOBBFKIXTSR
|
6.2 | IC50 | 3 | — | |
VNQBKUWYQVWGPY
|
6.2 | IC50 | 2 | — | |
WYCWXWHOPSRYNV
|
6.2 | IC50 | 2 | — | |
YUTIPCGWKBPNFQ
|
6.2 | IC50 | 2 | — | |
RCBNWWLBZCYILT
|
6.2 | IC50 | 5 | — | |
IVWMPAOBMMXESU
|
6.2 | IC50 | 5 | — | |
LODPWNVFWVRUDN
|
6.2 | IC50 | 6 | — | |
QSDVZPULRUJSBC
|
6.1 | Kd | 4 | — | |
YVBUTAWXLPEFFD
|
6.1 | IC50 | 5 | — | |
CICFFAJMTOTWDF
|
6.1 | IC50 | 5 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
SVSSPHFLEURYPE
|
6.1 | IC50 | 3 | — | |
BYTQGWNNPKNUGP
|
6.1 | IC50 | 2 | — | |
MYJVZDXYKKUBQF
|
6.1 | IC50 | 5 | — | |
PVYZELXSBIFXIA
|
6.1 | IC50 | 4 | — | |
CWWCJCDUPKPEJG
|
6.1 | IC50 | 4 | — | |
IICBFVCHOUCXJI
|
6.1 | IC50 | 5 | — | |
QSDVZPULRUJSBC
|
6.1 | Kd | 3 | — | |
BZYKWEQWEPHEQZ
|
6.1 | IC50 | 10 | Yes | |
GLWIEKCNAKUHPZ
|
6.0 | IC50 | 4 | — | |
NOCNKNHXOANVQW
|
6.0 | IC50 | 4 | — | |
PJPYMAJZJCYLKR
|
6.0 | IC50 | 3 | — | |
CKUSCWLPGIBNJZ
|
6.0 | IC50 | 4 | — | |
BCFGMOOMADDAQU
|
6.0 | Kd | 6 | Yes | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
NHHQJBCNYHBUSI
|
6.0 | Kd | 220 | — | |
VYXZSLJQQXROKX
|
6.0 | IC50 | 4 | — | |
CUIHSIWYWATEQL
|
6.0 | Kd | 61 | Yes | |
RERZXCUAKWVHPD
|
6.0 | IC50 | 4 | — | |
MABMRCWHKCPRMW
|
6.0 | IC50 | 5 | — | |
CBBGVZCNBLEQID
|
6.0 | IC50 | 5 | — | |
IPLZEFLYSZCVED
|
6.0 | IC50 | 2 | — | |
OPVRUFKBBKOABM
|
6.0 | IC50 | 4 | — | |
RTJQABCNNLMCJF
|
6.0 | IC50 | 3 | — | |
VWBMWDWXMHMJPH
|
6.0 | IC50 | 2 | — | |
ZYCQTLJPCIVXNL
|
6.0 | IC50 | 4 | — |