Target Details
| UniProt AC | Q9UBE8 |
|---|---|
| Gene Symbol | NLK |
| Protein Name | Serine/threonine-protein kinase NLK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 54
- Clinical molecules 10
- Avg pChEMBL 6.97
KEGG Pathways (4)
Active Molecules (54)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
8.9 | Kd | 599 | — | |
XCHWBXBDZRJVDP
|
8.6 | Ki | 51 | — | |
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
BHSOPYVVEZFHDB
|
8.4 | Ki | 25 | Yes | |
DKSNLQYRZJKYOC
|
8.3 | Ki | 51 | — | |
XYXLUJQBBIBJFV
|
8.3 | Ki | 36 | — | |
KKKRKRMVJRHDMG
|
8.2 | Kd | 14 | — | |
MWKSRKSEWLRPBL
|
7.8 | Kd | 1075 | — | |
XLFYOIVELARSKP
|
7.7 | Ki | 33 | — | |
ZXLFIHLBHMLHFJ
|
7.7 | Ki | 31 | — | |
DKZYXHCYPUVGAF
|
7.6 | Kd | 112 | — | |
CDMGBJANTYXAIV
|
7.6 | Kd | 34 | Yes | |
RWEHAHIEUDLKGT
|
7.6 | Ki | 33 | — | |
BLWQIEISIMYCHD
|
7.5 | Kd | 4 | — | |
QHKYPYXTTXKZST
|
7.5 | Kd | 28 | — | |
AHESYZXOYPHUOT
|
7.5 | Kd | 4 | — | |
ACNCCUVYXQGPKZ
|
7.5 | Ki | 31 | — | |
VAARYSWULJUGST
|
7.5 | Kd | 119 | Yes | |
UWDBNTXEKYRMSG
|
7.4 | Ki | 26 | — | |
ZFDGMDVYMNWICG
|
7.4 | IC50 | 10 | — | |
MADCXGNPDBWPLM
|
7.3 | Ki | 25 | — | |
QKPLUKMJEKRAJD
|
7.2 | Ki | 30 | Yes | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
LRLDYTTWQIFWBD
|
6.9 | Ki | 25 | — | |
FYSRKRZDBHOFAY
|
6.8 | Kd | 8 | — | |
ODPGGGTTYSGTGO
|
6.8 | Kd | 153 | — | |
CXQHYVUVSFXTMY
|
6.8 | Kd | 154 | — | |
JYYLVUFNAHSSFE
|
6.8 | Kd | 9 | — | |
SEJGTFPOEJWEGG
|
6.8 | Kd | 149 | — | |
HKSZLNNOFSGOKW
|
6.7 | Kd | 213 | — | |
QKNBRNSGPNCARD
|
6.6 | IC50 | 9 | — | |
RIUZPIBUSOHUKF
|
6.6 | Ki | 23 | — | |
ZBNZXTGUTAYRHI
|
6.6 | Kd | 102 | Yes | |
RKBYYWVZFBATHQ
|
6.5 | IC50 | 12 | — | |
FPWOHBGDJPLADA
|
6.5 | Kd | 4 | — | |
MTCHQDWUHQADSY
|
6.4 | Ki | 29 | — | |
VYPGLYMWNDRFGZ
|
6.4 | Kd | 12 | — | |
JUUFLLKHNYWHKP
|
6.3 | Kd | 12 | — | |
MFAQYJIYDMLAIM
|
6.3 | Kd | 130 | Yes | |
AUOSKLDNVNGKRR
|
6.3 | Kd | 6 | — | |
FQUBTLMSWPIBBP
|
6.2 | Kd | 4 | — | |
MLDQJTXFUGDVEO
|
6.2 | Kd | 85 | Yes | |
YULUHUJTIHWRMI
|
6.2 | Kd | 4 | — | |
GRKVQPWSPUXGKV
|
6.2 | Kd | 3 | — | |
CMJCXYNUCSMDBY
|
6.1 | Kd | 15 | — | |
ZUNCPEIOPMEIGV
|
6.1 | Kd | 4 | — | |
UIARLYUEJFELEN
|
6.1 | Kd | 289 | Yes | |
ZYQXEVJIFYIBHZ
|
6.1 | Kd | 5 | — | |
DCTBPIBEQFLAOQ
|
6.0 | Ki | 13 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |