Target Details
| UniProt AC | Q9UBE0 |
|---|---|
| Gene Symbol | SAE1 |
| Protein Name | SUMO-activating enzyme subunit 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00899 (ThiF) |
Summary
- Multi-target molecules 84
- Clinical molecules 0
- Avg pChEMBL 7.36
KEGG Pathways (1)
Active Molecules (84)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WMYZRWPUITZCPU
|
7.4 | IC50 | 2 | — | |
SPZOHGTXTGPSCS
|
7.4 | IC50 | 4 | — | |
JUVWGUHJFQQESY
|
7.3 | IC50 | 4 | — | |
XYUKAKFBAWCQRY
|
7.3 | IC50 | 4 | — | |
PLMYHNPIXAICML
|
7.3 | IC50 | 4 | — | |
VTYUOMASBKDZEV
|
7.2 | IC50 | 2 | — | |
PKHLGIWBWMPLAR
|
7.2 | IC50 | 4 | — | |
WMFPYJXJTLDGIG
|
7.2 | IC50 | 4 | — | |
WNCAZJJUZZNNAR
|
7.0 | IC50 | 2 | — | |
XKTWBXUBNVQZSI
|
7.0 | IC50 | 4 | — | |
IZYVMHSGDZFGFW
|
7.0 | IC50 | 4 | — | |
LXRZVMYMQHNYJB
|
7.0 | IC50 | 4 | — | |
FYCFHQRHVRHJML
|
6.9 | IC50 | 4 | — | |
QJRYTABJLBDESL
|
6.8 | IC50 | 2 | — | |
KNIHFXMFUCCLGH
|
6.4 | IC50 | 5 | — | |
HUSXUHAWHWEADE
|
6.3 | IC50 | 4 | — | |
CKMHTGNKKMADSO
|
6.3 | IC50 | 2 | — | |
DCIBEKBKAOZGMO
|
6.3 | IC50 | 3 | — | |
GCZZEBZXVDWJBN
|
6.3 | IC50 | 4 | — | |
GEVVUAXCPLJANF
|
6.3 | IC50 | 4 | — | |
OATWETZGGLHRAC
|
6.3 | IC50 | 2 | — | |
OVTMDKYPGLBLQS
|
6.2 | IC50 | 4 | — | |
AGBQKNBQESQNJD
|
6.2 | IC50 | 3 | — | |
WIKWWKTTXFVGLP
|
6.2 | IC50 | 2 | — | |
OHKMEPULKHPDSE
|
6.2 | IC50 | 2 | — | |
SPKHEQRHPVZIPW
|
6.2 | IC50 | 2 | — | |
ZJZDQWHYOGHGEQ
|
6.1 | IC50 | 2 | — | |
IDHVGLAGCDWRFN
|
6.1 | IC50 | 2 | — | |
BGYDUWHYSPAIGF
|
6.1 | IC50 | 3 | — | |
SZRJZDDPKYJEDA
|
6.1 | IC50 | 3 | — | |
ABIGPTDIQKRVCS
|
6.0 | IC50 | 4 | — | |
MZVDBDZUJDCBSC
|
6.0 | IC50 | 2 | — | |
WBVSZPHBBYURDY
|
6.0 | IC50 | 3 | — | |
ZCKFJAREHQZZOB
|
6.0 | IC50 | 4 | — |