Target Details
| UniProt AC | Q9QBY3 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype K (isolate 96CM-MP535) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 4
- Clinical molecules 0
- Avg pChEMBL 10.39
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ALWBGUNCNDFMFE
|
11.1 | Ki | 2 | — | |
KOYHHSRUNXTXFB
|
10.9 | Ki | 2 | — | |
CJBJHOAVZSMMDJ
|
10.6 | Ki | 3 | — | |
QMZQZXVEFMMDKK
|
8.9 | Ki | 2 | — |