Target Details
| UniProt AC | Q9P2K8 |
|---|---|
| Gene Symbol | EIF2AK4 |
| Protein Name | eIF-2-alpha kinase GCN2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12745 (HGTP_anticodon2) PF00069 (Pkinase) PF05773 (RWD) PF13393 (tRNA-synt_His) |
Summary
- Multi-target molecules 57
- Clinical molecules 8
- Avg pChEMBL 6.77
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NAVBCKMFEZHGEG
|
6.1 | IC50 | 2 | — | |
UPAHRQZYJXICAZ
|
6.1 | IC50 | 2 | — | |
ZRUJLUVFQVEJSE
|
6.1 | IC50 | 2 | — | |
QAEKSWBVYBVLNO
|
6.1 | IC50 | 5 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |