Target Details
| UniProt AC | Q9P2K8 |
|---|---|
| Gene Symbol | EIF2AK4 |
| Protein Name | eIF-2-alpha kinase GCN2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12745 (HGTP_anticodon2) PF00069 (Pkinase) PF05773 (RWD) PF13393 (tRNA-synt_His) |
Summary
- Multi-target molecules 57
- Clinical molecules 8
- Avg pChEMBL 6.77
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHHQJBCNYHBUSI
|
8.5 | Kd | 220 | — | |
UIARLYUEJFELEN
|
8.4 | Kd | 289 | Yes | |
QLCVZRYQHBSADC
|
8.3 | IC50 | 3 | — | |
ASGMFNBUXDJWJJ
|
8.1 | IC50 | 8 | — | |
LTKYUQAQPQMHNJ
|
8.0 | IC50 | 3 | — | |
JGQCTMHFTXGHEP
|
7.9 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 408 | — | |
ZZSBPGIGIUFJRA
|
7.8 | Kd | 46 | — | |
VAARYSWULJUGST
|
7.6 | Kd | 119 | Yes | |
KIGXQRBUVDDSPP
|
7.5 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 147 | Yes | |
YABJJWZLRMPFSI
|
7.3 | Kd | 34 | — | |
GUBJNPWVIUFSTR
|
7.1 | Kd | 103 | — | |
JWNPDZNEKVCWMY
|
7.0 | Kd | 57 | Yes | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
ITTRLTNMFYIYPA
|
6.8 | Kd | 17 | — | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
PIQCTGMSNWUMAF
|
6.6 | Kd | 137 | Yes | |
UBPYILGKFZZVDX
|
6.6 | Kd | 130 | Yes | |
PVNWAPAWLNSQHB
|
6.5 | IC50 | 2 | — | |
WVUNYSQLFKLYNI
|
6.5 | Kd | 46 | Yes | |
AETVLBTWUVIWCA
|
6.5 | IC50 | 2 | — | |
BDYQIMPHYQJENY
|
6.5 | IC50 | 2 | — | |
BEMXOHYKXHMKOY
|
6.5 | IC50 | 2 | — | |
BLLYYAVGBOPRJI
|
6.5 | IC50 | 2 | — | |
DEQZEUDASDTSSV
|
6.5 | IC50 | 2 | — | |
FIYYRTKUHIMARG
|
6.5 | IC50 | 2 | — | |
IRINBZJIFSYGRV
|
6.5 | IC50 | 2 | — | |
KYIIDZUSEBPYMT
|
6.5 | IC50 | 2 | — | |
MGLXTGHVERCWAN
|
6.5 | IC50 | 2 | — | |
NRYBQVQBNOQOAV
|
6.5 | IC50 | 2 | — | |
PDVKNBJHJMVTOD
|
6.5 | IC50 | 2 | — | |
RDPSDALZCPLTHI
|
6.5 | IC50 | 2 | — | |
RSZWKPZDKYYNBU
|
6.5 | IC50 | 2 | — | |
SVGIOLWOWDFKCI
|
6.5 | IC50 | 2 | — | |
SYDJLQGRTCATIS
|
6.5 | IC50 | 2 | — | |
UTYJZDXOURRFAS
|
6.5 | IC50 | 2 | — | |
UWVVESMKNHRLBR
|
6.5 | IC50 | 2 | — | |
VJGYCLGKKGWXLJ
|
6.5 | IC50 | 2 | — | |
VZFZJDBCZWELMK
|
6.5 | IC50 | 2 | — | |
WBXCQVZFFNMQEM
|
6.5 | IC50 | 2 | — | |
XRIHVFZLYWJMPM
|
6.5 | IC50 | 2 | — | |
YICGALUZBYPKNW
|
6.5 | IC50 | 2 | — | |
ZSXYTEMLUYJFEY
|
6.5 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
NYVUSSXLPQHLMH
|
6.4 | IC50 | 3 | — | |
HHCBMISMPSAZBF
|
6.3 | IC50 | 23 | — | |
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
AQCKYYPUJQXLJN
|
6.1 | IC50 | 2 | — | |
CVMXSGAHYHKSJR
|
6.1 | IC50 | 2 | — |