Target Details
| UniProt AC | Q9P2J5 |
|---|---|
| Gene Symbol | LARS1 |
| Protein Name | Leucine--tRNA ligase, cytoplasmic |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08264 (Anticodon_1) PF24810 (RBD_LARS1) PF00133 (tRNA-synt_1) PF22947 (ULD_3) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FREGHQKQLWGWHX
|
8.2 | IC50 | 2 | — | |
YABWOCJHKKFQIN
|
7.8 | IC50 | 3 | — | |
XFEDFDTWJLGMBO
|
7.7 | IC50 | 2 | — | |
FDKDOHYGEOEKBT
|
7.5 | IC50 | 2 | — | |
JTTTWNOSNPJPPL
|
6.8 | IC50 | 2 | — | |
YLOJPCMXCBVFGR
|
6.7 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
6.6 | Kd | 1075 | — | |
NBOMIQZITNLNJQ
|
6.3 | IC50 | 2 | — | |
FUNOATJOTYEZJZ
|
6.1 | IC50 | 2 | — | |
NAKYNJKKYDJABY
|
6.1 | IC50 | 2 | — | |
BIRNJUNFRITRFT
|
6.0 | IC50 | 2 | — |