Target Details
| UniProt AC | Q9P286 |
|---|---|
| Gene Symbol | PAK5 |
| Protein Name | Serine/threonine-protein kinase PAK 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 23
- Clinical molecules 7
- Avg pChEMBL 7.01
KEGG Pathways (9)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.9 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
8.6 | Kd | 408 | — | |
KGPGFQWBCSZGEL
|
8.1 | Kd | 59 | Yes | |
FPQNRXITKTZFMF
|
7.9 | Kd | 13 | — | |
RTGFZUPLFGBDKE
|
7.8 | IC50 | 2 | — | |
AYCPARAPKDAOEN
|
7.7 | IC50 | 73 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
7.3 | Kd | 170 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
DGLFSNZWRYADFC
|
7.0 | IC50 | 12 | — | |
RZXMIHOUHYSGJO
|
6.9 | IC50 | 4 | — | |
TXGKRVFSSHPBAJ
|
6.8 | IC50 | 11 | — | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
MFAQYJIYDMLAIM
|
6.3 | Kd | 130 | Yes | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
KDKUVYLMPJIGKA
|
6.1 | Kd | 91 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |