Target Details
| UniProt AC | Q9P1W9 |
|---|---|
| Gene Symbol | PIM2 |
| Protein Name | Serine/threonine-protein kinase pim-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,276
- Clinical molecules 10
- Avg pChEMBL 7.77
KEGG Pathways (2)
Active Molecules (2,276)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BUSRDZKIQOWUOO
|
8.8 | IC50 | 3 | — | |
CUEWSGPOORVNOX
|
8.8 | IC50 | 2 | — | |
DWJRVXUXEZICSB
|
8.8 | IC50 | 3 | — | |
KRXHIAQHNCEJEE
|
8.8 | IC50 | 3 | — | |
ROWCDUKNAFYOMJ
|
8.8 | IC50 | 3 | — | |
VLOSGHYSCVRVJH
|
8.8 | IC50 | 2 | — | |
ZBIYVIOSDQBGRR
|
8.8 | IC50 | 3 | — | |
DFRBAIKCWZMMMO
|
8.8 | IC50 | 3 | — | |
FUOLJDPZDKQMEX
|
8.8 | IC50 | 2 | — | |
LMYCHBCZOYRSRO
|
8.8 | Ki | 3 | — | |
BZUBDLKATGBRRF
|
8.8 | IC50 | 2 | — | |
CYOQMLSODZDBGH
|
8.8 | Ki | 3 | — | |
IDHYALMZKJRNKP
|
8.8 | IC50 | 2 | — | |
OAVGBZOFDPFGPJ
|
8.8 | Ki | 42 | Yes | |
YAJGELPVDBECTQ
|
8.8 | IC50 | 2 | — | |
ACDKOFBRGHETMP
|
8.8 | IC50 | 2 | — | |
MAODNWJWGVULBD
|
8.8 | IC50 | 3 | — | |
QDBBFQPBTRDBMD
|
8.8 | IC50 | 2 | — | |
KYXJMCQQNZDWIT
|
8.8 | IC50 | 3 | — | |
MZEDYGZPEWMQOQ
|
8.8 | Ki | 3 | — | |
FHAPDLVADXCIGY
|
8.8 | Ki | 3 | — | |
GAMSTIVHSDPIFY
|
8.8 | Ki | 3 | — | |
MHBGRNASPWNGMV
|
8.8 | Ki | 3 | — | |
OHWHNLRNFFGOSF
|
8.8 | IC50 | 3 | — | |
QGQNOAJYKWNLCF
|
8.8 | IC50 | 3 | — | |
SMYZVTZPMXEMEO
|
8.8 | IC50 | 2 | — | |
VGTXZFMBNSOWGX
|
8.8 | IC50 | 3 | — | |
WSBXTXMVHFPAPA
|
8.8 | IC50 | 3 | — | |
KTOADPOSUJJLPI
|
8.8 | IC50 | 3 | — | |
LBSWUVMKCABART
|
8.8 | Ki | 3 | — | |
NWDVLGCDUFSSHA
|
8.8 | IC50 | 3 | — | |
RRSYIVJLGUPYPY
|
8.8 | IC50 | 2 | — | |
KWQWZDJFPORDSD
|
8.8 | IC50 | 2 | — | |
LPJZLEGMOKXVFB
|
8.8 | IC50 | 3 | — | |
NYMXZZBYJOQYQM
|
8.8 | IC50 | 3 | — | |
BMRHAWSJNXXRJI
|
8.7 | IC50 | 2 | — | |
CMCGBWKSQYENCR
|
8.7 | IC50 | 2 | — | |
JXTNSWUVLITLAJ
|
8.7 | IC50 | 2 | — | |
OLQLOEJZYFROOC
|
8.7 | IC50 | 2 | — | |
PNJLKNVXTURZGB
|
8.7 | IC50 | 2 | — | |
XKCUAIJHVDEELV
|
8.7 | Ki | 3 | — | |
FBUGFYYXGPZIKL
|
8.7 | IC50 | 2 | — | |
LGIGKYXJCHINMH
|
8.7 | IC50 | 3 | — | |
UMSZCQJFRUIBCG
|
8.7 | Ki | 3 | — | |
HKSZLNNOFSGOKW
|
8.7 | Kd | 213 | — | |
JJHPKDPBGCWUNR
|
8.7 | IC50 | 2 | — | |
PJGYOXBIUJBVPM
|
8.7 | IC50 | 3 | — | |
RRSYIVJLGUPYPY
|
8.7 | IC50 | 2 | — | |
UGSZUXSPYQGPRH
|
8.7 | IC50 | 2 | — | |
WDZRXBBDZLKEFS
|
8.7 | IC50 | 3 | — |