Target Details
| UniProt AC | Q9P1W9 |
|---|---|
| Gene Symbol | PIM2 |
| Protein Name | Serine/threonine-protein kinase pim-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,276
- Clinical molecules 10
- Avg pChEMBL 7.77
KEGG Pathways (2)
Active Molecules (2,276)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHYXMWPAQOHZQD
|
8.0 | IC50 | 3 | — | |
NJPWCTYVEJIQBM
|
8.0 | Ki | 72 | — | |
RVEDMOLIJBWGQX
|
8.0 | Ki | 3 | — | |
SHYCQJRIHDQKDV
|
8.0 | IC50 | 4 | — | |
STWDLMHONRHMTF
|
8.0 | IC50 | 3 | — | |
SXGXDOZGWJTWBA
|
8.0 | IC50 | 3 | — | |
VHAIPPXUMKWXIR
|
8.0 | IC50 | 2 | — | |
VSYLYSOTCDFRSM
|
8.0 | IC50 | 2 | — | |
VXYDJXMHISGSDA
|
8.0 | Ki | 59 | — | |
WLBVZYXAXNRNOX
|
8.0 | Ki | 3 | — | |
WSADVDPLODZOTP
|
8.0 | IC50 | 2 | — | |
ZNTIFAHOYOIGGK
|
8.0 | IC50 | 3 | — | |
BLHWEGXFMWEIHN
|
8.0 | IC50 | 3 | — | |
GDXMDKRKEIKPLW
|
8.0 | IC50 | 3 | — | |
LRVOQVWUCGGLLL
|
8.0 | IC50 | 2 | — | |
VJXUXTWQBIILQL
|
8.0 | Ki | 3 | — | |
CPVVGAAUXSVJPE
|
8.0 | Ki | 3 | — | |
CWVPFBCGDKVIPY
|
8.0 | Ki | 3 | — | |
DSFJTSSJSJDOGO
|
8.0 | IC50 | 2 | — | |
IIYNOYBNJALAMM
|
8.0 | IC50 | 3 | — | |
NIRJXKZEFQTBIC
|
8.0 | IC50 | 2 | — | |
QBMHBUSZNODSPS
|
8.0 | Ki | 3 | — | |
SDHRADPEFDLIKD
|
8.0 | IC50 | 3 | — | |
UJBRJYXRVHBJQM
|
8.0 | IC50 | 2 | — | |
UTNCOKVXILEJCJ
|
8.0 | IC50 | 2 | — | |
AUSOZFFBBXRILI
|
8.0 | Ki | 3 | — | |
CHFXZLZGCMQMBM
|
8.0 | IC50 | 3 | — | |
KSUJTDNWWVQOFC
|
8.0 | Ki | 3 | — | |
PAWVEZOTRVPHRU
|
8.0 | IC50 | 2 | — | |
RJQJFTUVYNAFRC
|
8.0 | IC50 | 2 | — | |
SUYTXTNWGWYQEV
|
8.0 | IC50 | 2 | — | |
WCLBXMSWYPPACJ
|
8.0 | IC50 | 3 | — | |
ATEORQMBWPIYQV
|
8.0 | IC50 | 3 | — | |
BQHHQEYEYHRNQA
|
8.0 | IC50 | 2 | — | |
CSYNBNGKBZGJAV
|
8.0 | IC50 | 3 | — | |
GIHUWFBQWLLTIZ
|
8.0 | IC50 | 4 | — | |
JXVXKOPUJQFJEO
|
8.0 | Ki | 3 | — | |
LQASHUDUJOBHMP
|
8.0 | IC50 | 3 | — | |
PKGOHWVMPQTAGB
|
8.0 | IC50 | 2 | — | |
QBDOORMZDCRUOU
|
8.0 | IC50 | 3 | — | |
SMFLEXPDEWVLCB
|
8.0 | IC50 | 2 | — | |
TVKZQOKEZKIHAL
|
8.0 | IC50 | 3 | — | |
UEPZXHSQXVBLNH
|
8.0 | IC50 | 2 | — | |
UOMPPOVQMYNXST
|
8.0 | IC50 | 2 | — | |
WWECFSFDKPKNDT
|
8.0 | IC50 | 3 | — | |
WXBFQEMPNLLMNB
|
8.0 | Ki | 3 | — | |
XUGBYZKANWTVIN
|
8.0 | IC50 | 2 | — | |
AYNCNNOVAOFEMG
|
8.0 | IC50 | 3 | — | |
ANPJHKVBDUXPEB
|
7.9 | IC50 | 2 | — | |
KDRBBKILEOZBCW
|
7.9 | IC50 | 2 | — |