Target Details
| UniProt AC | Q9P1W9 |
|---|---|
| Gene Symbol | PIM2 |
| Protein Name | Serine/threonine-protein kinase pim-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,276
- Clinical molecules 10
- Avg pChEMBL 7.77
KEGG Pathways (2)
Active Molecules (2,276)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FPBWUTAWSOLPQI
|
9.9 | Ki | 3 | — | |
SVYHADKWCWQANW
|
9.9 | Ki | 3 | — | |
JTYPMPKUWKZGBR
|
9.9 | IC50 | 2 | — | |
ZQNLSYAFNSXFET
|
9.9 | IC50 | 2 | — | |
URJWEBIIRXSJGD
|
9.9 | IC50 | 2 | — | |
APJNEWHEOPKPSA
|
9.8 | Ki | 3 | — | |
BAUZKJYZGGFFLL
|
9.8 | Ki | 3 | — | |
KFEFAUXTDOPDKJ
|
9.8 | IC50 | 2 | — | |
MDSSZYNUYNBVFZ
|
9.8 | IC50 | 2 | — | |
NMBLJOILHIVHIT
|
9.8 | IC50 | 2 | — | |
SGCVXQAEURWEAZ
|
9.8 | IC50 | 2 | — | |
UMICCZFMUZBZJG
|
9.8 | IC50 | 2 | — | |
NDQPAYWKSVOGPA
|
9.8 | IC50 | 2 | — | |
JEVIKKKBDOXJFA
|
9.8 | Ki | 3 | — | |
PAKQZSJYQOIVOH
|
9.8 | Ki | 3 | — | |
QJYRTBVKAJEXQS
|
9.8 | IC50 | 2 | — | |
ZNOTUHKIYPIPHI
|
9.8 | Ki | 3 | — | |
PPKOMRSAECKGDB
|
9.8 | IC50 | 2 | — | |
AWSQCMGUEHCTJL
|
9.7 | IC50 | 2 | — | |
LBUJNZMSBAMNNW
|
9.7 | IC50 | 2 | — | |
XIXPZKIRXUHXDD
|
9.7 | IC50 | 2 | — | |
AQFQLFWVDMMENJ
|
9.7 | Ki | 3 | — | |
UOJNFBQURVKKJP
|
9.7 | IC50 | 2 | — | |
IWGQMHPNGOJNRQ
|
9.7 | IC50 | 2 | — | |
NDXAAESWIVMHKZ
|
9.7 | IC50 | 2 | — | |
ZUJJFZSSMJANFF
|
9.7 | IC50 | 2 | — | |
ASZCABSVZBJTKA
|
9.7 | IC50 | 3 | — | |
GPGQKMLTKINISD
|
9.7 | IC50 | 2 | — | |
IKFWWTFURAIGPU
|
9.7 | Ki | 3 | — | |
ISSQSUGBRMTNBJ
|
9.7 | IC50 | 3 | — | |
LBUJNZMSBAMNNW
|
9.7 | IC50 | 2 | — | |
MLAWVMHISKOVHW
|
9.7 | IC50 | 3 | — | |
OSBCYEMTQYPIMH
|
9.7 | Ki | 3 | — | |
WFTRLROTBYTPTM
|
9.7 | IC50 | 2 | — | |
XFUKFDJFEAQRRG
|
9.7 | Ki | 3 | — | |
XNTIENONSOGMRS
|
9.7 | IC50 | 2 | — | |
YAJGELPVDBECTQ
|
9.7 | IC50 | 3 | — | |
YMMNFBQYTKNEGM
|
9.7 | Ki | 3 | — | |
YWQCLSBVOVPANW
|
9.7 | IC50 | 2 | — | |
YBENUWLHUXAJFZ
|
9.7 | Ki | 3 | — | |
PPKOMRSAECKGDB
|
9.7 | IC50 | 2 | — | |
LQILNMFAVKTKBG
|
9.7 | IC50 | 2 | — | |
AZUDXPDVDQXJJH
|
9.6 | Ki | 3 | — | |
OIZRMKSUYVZCDN
|
9.6 | Ki | 3 | — | |
UZSKGLPUMSUOBY
|
9.6 | Ki | 3 | — | |
WLKLBBSKBUEHCT
|
9.6 | IC50 | 2 | — | |
AFPFWSQRRIQPHP
|
9.6 | Ki | 3 | — | |
IOOVJBGMLHBOOX
|
9.6 | IC50 | 2 | — | |
OIZRMKSUYVZCDN
|
9.6 | Ki | 3 | — | |
SWVVEDSPZBMVBS
|
9.6 | IC50 | 2 | — |