Target Details
| UniProt AC | Q9P1W9 |
|---|---|
| Gene Symbol | PIM2 |
| Protein Name | Serine/threonine-protein kinase pim-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,276
- Clinical molecules 10
- Avg pChEMBL 7.77
KEGG Pathways (2)
Active Molecules (2,276)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJBLYAOGZIACGS
|
11.4 | Ki | 3 | — | |
KMIKZMJCDRKNJE
|
11.2 | Ki | 3 | — | |
GAPPKQMJLOBLDJ
|
10.7 | IC50 | 3 | — | |
VRQXRVAKPDCRCI
|
10.7 | IC50 | 3 | — | |
NJOKRJWJYGYTRB
|
10.7 | IC50 | 2 | — | |
BEXSRDRFSVXXPU
|
10.5 | Ki | 3 | — | |
DWZMCUJAYLNSOB
|
10.4 | IC50 | 2 | — | |
IBNILFRNVFTCBR
|
10.4 | IC50 | 2 | — | |
TWIFKBILIHXMMI
|
10.4 | Ki | 3 | — | |
DVKOJQHRIKGCMQ
|
10.4 | IC50 | 2 | — | |
QVQNZMJSTKPJKL
|
10.4 | IC50 | 2 | — | |
GZHPOGVPEBAKBW
|
10.4 | Ki | 3 | — | |
OJACGGVADSBVKM
|
10.4 | IC50 | 2 | — | |
XCEBXSIYXWIQPP
|
10.4 | Ki | 3 | — | |
HNGYLMVBNQDLKS
|
10.3 | IC50 | 2 | — | |
DXFVPMMMQNXSOZ
|
10.3 | Ki | 3 | — | |
DDQXBYGNFGPJRL
|
10.3 | IC50 | 3 | — | |
MLAWVMHISKOVHW
|
10.3 | IC50 | 3 | — | |
VHHMNEWIYJHDIY
|
10.3 | Ki | 3 | — | |
WPKXXVMGORDACP
|
10.3 | IC50 | 2 | — | |
UWSPFENPUCOTKU
|
10.2 | IC50 | 2 | — | |
SMKDKOFQQMLFPP
|
10.2 | IC50 | 3 | — | |
UXRGJORUNNVPFQ
|
10.1 | IC50 | 2 | — | |
VKNMCBUJJJKJQM
|
10.1 | Ki | 3 | — | |
BRUNMKAHHCQBLZ
|
10.1 | IC50 | 2 | — | |
CTADVIUFFUGUBU
|
10.1 | IC50 | 2 | — | |
OYVCFKLZLLYNOW
|
10.1 | Ki | 3 | — | |
ASZCABSVZBJTKA
|
10.1 | IC50 | 3 | — | |
BHBIGGOODMPQTA
|
10.1 | IC50 | 2 | — | |
RLVXEHCCQLTFMJ
|
10.1 | IC50 | 2 | — | |
XWOSSDMMJDYDBX
|
10.1 | Ki | 3 | — | |
GEYAXZBDDHIAPF
|
10.1 | IC50 | 3 | — | |
UCLIZEJSCGLLJP
|
10.0 | Ki | 3 | — | |
FPIJQPCUMVUNOE
|
10.0 | IC50 | 2 | — | |
VFYCNKMVBINXBE
|
10.0 | IC50 | 2 | — | |
AENSKLYNJAPICQ
|
10.0 | IC50 | 2 | — | |
GTKNYUJNLDGSDF
|
10.0 | IC50 | 3 | — | |
HPFPEYFODXCUDT
|
10.0 | IC50 | 2 | — | |
JEVIKKKBDOXJFA
|
10.0 | Ki | 3 | — | |
LDCFHYFYINOQIH
|
10.0 | IC50 | 2 | — | |
NHXVGMQFCYBLTL
|
10.0 | Ki | 8 | — | |
OLFGXMCJTMYBMY
|
10.0 | IC50 | 2 | — | |
PCKUZAUQQUCSJT
|
10.0 | IC50 | 2 | — | |
XKEPASMYHMOCPP
|
10.0 | IC50 | 3 | — | |
ADHFWXANXDIZPQ
|
10.0 | Ki | 3 | — | |
GPGQKMLTKINISD
|
10.0 | IC50 | 3 | — | |
KFEFAUXTDOPDKJ
|
10.0 | IC50 | 2 | — | |
ZMLWOFMZTHIIIJ
|
10.0 | IC50 | 2 | — | |
OHXQPUAQXWTIOM
|
9.9 | Ki | 3 | — | |
CBXHYUCLQVWOJZ
|
9.9 | IC50 | 2 | — |