Target Details
| UniProt AC | Q9P0L2 |
|---|---|
| Gene Symbol | MARK1 |
| Protein Name | Serine/threonine-protein kinase MARK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 23
- Clinical molecules 7
- Avg pChEMBL 7.05
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.4 | IC50 | 408 | — | |
OFIFLUFVENTCNZ
|
8.7 | IC50 | 11 | — | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
HKSZLNNOFSGOKW
|
8.4 | Kd | 213 | — | |
NXSJMRCTGYTSTK
|
8.1 | Kd | 200 | — | |
UKBGBACORPRCGG
|
7.6 | IC50 | 17 | — | |
QQWUGDVOUVUTOY
|
7.5 | Kd | 231 | Yes | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
TZOLUHQWLXJGBH
|
7.0 | IC50 | 7 | Yes | |
XVBWTZHNQZHFHR
|
6.9 | IC50 | 5 | — | |
AILRADAXUVEEIR
|
6.9 | IC50 | 75 | — | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 91 | Yes | |
AXWDQRXGOKDXJT
|
6.7 | Kd | 6 | — | |
NHHQJBCNYHBUSI
|
6.6 | Kd | 220 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
FWLMVFUGMHIOAA
|
6.3 | IC50 | 26 | — | |
PLZWVXKEQYGKTJ
|
6.2 | IC50 | 7 | Yes | |
KDKUVYLMPJIGKA
|
6.2 | Kd | 91 | Yes | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |