Target Details
| UniProt AC | Q9P0G3 |
|---|---|
| Gene Symbol | KLK14 |
| Protein Name | Kallikrein-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 25
- Clinical molecules 0
- Avg pChEMBL 7.0
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PJWRVDWTVAOOQV
|
9.4 | Ki | 7 | — | |
ZXLZUCADFTVDHK
|
8.9 | Ki | 3 | — | |
VRMZLUPLYRHORK
|
8.7 | Ki | 6 | — | |
AOMZQHHLSHFCGW
|
8.2 | Ki | 2 | — | |
RDZNGZAQRWVXQR
|
7.7 | Ki | 2 | — | |
SXIFJSHGLQMOET
|
7.6 | Ki | 3 | — | |
NWAGTUQRZPXSNY
|
7.5 | IC50 | 6 | — | |
WICLAAAUGCVLKH
|
7.1 | Ki | 2 | — | |
JTQBMTFVGGUDPN
|
7.0 | Ki | 3 | — | |
WYFUNPGYPSDKCF
|
7.0 | Ki | 3 | — | |
NWAGTUQRZPXSNY
|
6.9 | IC50 | 5 | — | |
STJCUZOTQPIXIR
|
6.8 | Ki | 2 | — | |
MICLUGCMNGFNIQ
|
6.8 | IC50 | 3 | — | |
OCOZTJLWHRDAJG
|
6.7 | IC50 | 4 | — | |
QFJOOWSJASQPAX
|
6.6 | IC50 | 7 | — | |
OPVLRSNIYJHUNK
|
6.5 | IC50 | 4 | — | |
ATSZLVKWSVRBLA
|
6.4 | IC50 | 4 | — | |
NWAGTUQRZPXSNY
|
6.4 | IC50 | 4 | — | |
KTPYVEWDDQSBAX
|
6.3 | Ki | 5 | — | |
WLGDDLRHBMVFMQ
|
6.3 | Ki | 3 | — | |
FKSBHSQGFGGOEF
|
6.1 | Ki | 4 | — | |
YENXZRUMZHNJKP
|
6.1 | IC50 | 4 | — | |
IDFLVSYGEYZZGR
|
6.0 | IC50 | 4 | — | |
MRAAINIKTLQAMC
|
6.0 | IC50 | 4 | — | |
UNPMSHQAFOCFFH
|
6.0 | Ki | 3 | — |