Target Details
| UniProt AC | Q9NZJ5 |
|---|---|
| Gene Symbol | EIF2AK3 |
| Protein Name | Eukaryotic translation initiation factor 2-alpha kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 154
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (11)
Associated Diseases (1)
Active Molecules (154)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KWZXRCBCAYLKPI
|
9.7 | IC50 | 3 | — | |
SIXVRXARNAVBTC
|
9.4 | IC50 | 12 | — | |
QAEKSWBVYBVLNO
|
9.3 | IC50 | 5 | — | |
OTGQMOPRPFKJKL
|
9.1 | IC50 | 3 | — | |
YNDQMKBAYRFBMW
|
8.7 | IC50 | 2 | — | |
CVTISFUIJNOONP
|
8.5 | IC50 | 2 | — | |
GZISLAWEFNWGCT
|
8.5 | IC50 | 2 | — | |
ZAEWPVUVQVUGEE
|
8.5 | IC50 | 2 | — | |
PPJWJOYOOLVOPL
|
8.4 | IC50 | 2 | — | |
BRIWRAFDHZTJPE
|
8.4 | IC50 | 2 | — | |
PVNWAPAWLNSQHB
|
8.4 | IC50 | 2 | — | |
XMXNMDQZYHHSSJ
|
8.4 | IC50 | 2 | — | |
VWKOZUNKVKWHGC
|
8.4 | IC50 | 2 | — | |
PRWSIEBRGXYXAJ
|
8.3 | IC50 | 4 | — | |
VJSNNBDPTLXPPT
|
8.3 | IC50 | 2 | — | |
XHUVPVATWTZPPU
|
8.2 | IC50 | 2 | — | |
LIGGMBSSOOVGAE
|
8.2 | IC50 | 2 | — | |
WFLLOUGNTSBEON
|
8.1 | IC50 | 2 | — | |
FYRWUAWBPDXQPZ
|
8.1 | IC50 | 2 | — | |
JSHFTMAPLMJGCF
|
8.1 | IC50 | 2 | — | |
HFOKVVVCWLIUBP
|
8.0 | IC50 | 3 | — | |
VYZYOJULVVGQRS
|
8.0 | IC50 | 2 | — | |
OYPSWGQEIRWPRG
|
8.0 | IC50 | 2 | — | |
XMJPZNCMRRFABT
|
7.8 | IC50 | 2 | — | |
MFJJLZIXKPDJHY
|
7.8 | IC50 | 2 | — | |
LBLBTNIBKKNQAH
|
7.8 | IC50 | 2 | — | |
PZUHKQRSUMVMFJ
|
7.7 | IC50 | 2 | — | |
VNDDOAWIHYNTOI
|
7.7 | IC50 | 3 | — | |
YXMQYIZUPKQHRP
|
7.7 | IC50 | 2 | — | |
JTSYRPMZSWPUHL
|
7.7 | IC50 | 2 | — | |
PNRYWGAXPBKWAG
|
7.6 | IC50 | 2 | — | |
BRIWRAFDHZTJPE
|
7.6 | IC50 | 2 | — | |
RPSNLKRQONAZHZ
|
7.6 | IC50 | 2 | — | |
VLZBNNUEXCARSV
|
7.5 | IC50 | 2 | — | |
XNYZWJDKGDUFBJ
|
7.5 | IC50 | 2 | — | |
XFMJNFJUBNDIMV
|
7.5 | IC50 | 2 | — | |
FBFPWPVDVUHEKP
|
7.5 | IC50 | 2 | — | |
RIBDKTGIOVNZBA
|
7.5 | IC50 | 2 | — | |
JPGLGZVWXAXTCH
|
7.5 | IC50 | 2 | — | |
AHLQDZCJPCLDJM
|
7.4 | IC50 | 2 | — | |
SIKKESBUGBWVRF
|
7.4 | IC50 | 3 | — | |
CUTMOOSDQSRDHK
|
7.3 | IC50 | 2 | — | |
WCBNKFWTMBJQOT
|
7.3 | IC50 | 2 | — | |
YCRNZPYPOFXDCB
|
7.3 | IC50 | 2 | — | |
KEBPJQMTPGEFMC
|
7.3 | IC50 | 2 | — | |
FNPGBBNIHLCSGJ
|
7.3 | IC50 | 2 | — | |
NQCYZSVEYSASFG
|
7.3 | IC50 | 2 | — | |
PGKOVECYHRNFSL
|
7.3 | IC50 | 2 | — | |
UOICEVZJMJOXIJ
|
7.3 | IC50 | 2 | — | |
YEPKWUFXXCZRIE
|
7.3 | IC50 | 2 | — |