Target Details
| UniProt AC | Q9NZ42 |
|---|---|
| Gene Symbol | PSENEN |
| Protein Name | Gamma-secretase subunit PEN-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10251 (PEN-2) |
Summary
- Multi-target molecules 1,927
- Clinical molecules 1
- Avg pChEMBL 7.37
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (1,927)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DSWLPEPFDLVFLT
|
7.7 | IC50 | 6 | — | |
FIJKEHHUIPTQRA
|
7.7 | IC50 | 6 | — | |
WOOMNCKEYUWJFD
|
7.7 | IC50 | 6 | — | |
ZVZKSTFCROUTRV
|
7.7 | IC50 | 6 | — | |
ACFIVGINFPMMJL
|
7.7 | IC50 | 6 | — | |
COQZVNPOYIUIIK
|
7.7 | IC50 | 6 | — | |
FRZXDSUPCFEKPH
|
7.7 | IC50 | 6 | — | |
GBIIFFGTDHZPKQ
|
7.7 | IC50 | 6 | — | |
GGTOKLPPMHMCOK
|
7.7 | IC50 | 6 | — | |
HFJZRWCWCVNTKK
|
7.7 | IC50 | 6 | — | |
IBWCDWOKROYSDN
|
7.7 | IC50 | 6 | — | |
MWURKMXQKGEUQZ
|
7.7 | IC50 | 6 | — | |
PEJUJRISYADBIN
|
7.7 | IC50 | 6 | — | |
RDPXIFBTABKBRO
|
7.7 | IC50 | 6 | — | |
RGCLCQZLVUNQPT
|
7.7 | IC50 | 6 | — | |
SACXAYXNJDLYGA
|
7.7 | IC50 | 6 | — | |
SAQXZEFKPJEJJL
|
7.7 | IC50 | 6 | — | |
SKKNGTJHVDVDQB
|
7.7 | IC50 | 6 | — | |
SOORDTTXOIHQDM
|
7.7 | IC50 | 6 | — | |
WVTRPWCJXUGFFA
|
7.7 | IC50 | 6 | — | |
ZFSPCKGRLFLVFF
|
7.7 | IC50 | 6 | — | |
ZVJWWQYNYFOGEZ
|
7.7 | IC50 | 6 | — | |
BLNOHOHTYGWWGU
|
7.7 | IC50 | 6 | — | |
COUFGTNLBNJCIM
|
7.7 | IC50 | 6 | — | |
GVZWJBACHKMERR
|
7.7 | IC50 | 6 | — | |
HIZHNHITDDKGGY
|
7.7 | IC50 | 6 | — | |
IOWRLBKYIIYWKF
|
7.7 | IC50 | 6 | — | |
IVHPMGRSWKGUQU
|
7.7 | IC50 | 6 | — | |
QRNBVQVYYYFGKJ
|
7.7 | IC50 | 7 | — | |
SBIKCUDPZRLNAC
|
7.7 | IC50 | 6 | — | |
SBPPZYYVSLBSSX
|
7.7 | IC50 | 6 | — | |
WRUHKVPKXIJRIY
|
7.7 | IC50 | 6 | — | |
ZVMAHZWUDYKAJT
|
7.7 | IC50 | 6 | — | |
BCIWPZDEVCOVHV
|
7.7 | IC50 | 6 | — | |
JCCTVKXXDWBDOU
|
7.7 | IC50 | 6 | — | |
AGUUKVAZOCMGFC
|
7.7 | IC50 | 6 | — | |
FVGUKPOYBXSMGS
|
7.7 | IC50 | 6 | — | |
GOWXCQHLZOLDPC
|
7.7 | IC50 | 6 | — | |
HGFAJEPTMZEYKW
|
7.7 | IC50 | 6 | — | |
JDKUGBDQALUAPJ
|
7.7 | IC50 | 6 | — | |
MABHMOXKRMWJGK
|
7.7 | IC50 | 6 | — | |
MTPJBVCVEZMXMP
|
7.7 | IC50 | 6 | — | |
OOBIJSQKFMWPBV
|
7.7 | IC50 | 6 | — | |
TXILJKJKOYLCFT
|
7.7 | IC50 | 6 | — | |
ZPMAVVZDYBVVFM
|
7.7 | IC50 | 6 | — | |
HBENWAJEVNKJSM
|
7.7 | IC50 | 6 | — | |
HXLYXVBIWJFTFT
|
7.7 | IC50 | 7 | — | |
FRKVPKQQZQNZHG
|
7.6 | IC50 | 6 | — | |
HVSDODQLRPYGML
|
7.6 | IC50 | 6 | — | |
JMFPNAQZNGBMQY
|
7.6 | IC50 | 6 | — |