Target Details
| UniProt AC | Q9NZ08 |
|---|---|
| Gene Symbol | ERAP1 |
| Protein Name | Endoplasmic reticulum aminopeptidase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11838 (ERAP1_C) PF01433 (Peptidase_M1) PF17900 (Peptidase_M1_N) |
Summary
- Multi-target molecules 30
- Clinical molecules 0
- Avg pChEMBL 6.66
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JEQPENJEYBAHIE
|
7.5 | IC50 | 3 | — | |
QKFOTLXPIIESQI
|
7.5 | IC50 | 5 | — | |
FLHXMLUIEURZLV
|
7.4 | IC50 | 3 | — | |
QCPJTEUURKCRNT
|
7.4 | IC50 | 4 | — | |
QJVIFKMCLOJOGV
|
7.3 | IC50 | 3 | — | |
GSWUIYHGTPVQDP
|
7.2 | IC50 | 3 | — | |
ASBAZJSDHGVMRZ
|
7.2 | IC50 | 3 | — | |
WWZWLDVQUBJSGD
|
7.0 | IC50 | 3 | — | |
WVARWRXWGWJNRJ
|
7.0 | IC50 | 3 | — | |
GXEDNWSUKCJLLB
|
7.0 | IC50 | 3 | — | |
YNFZCLOZANIMIN
|
6.9 | IC50 | 3 | — | |
QWLYILUODIZPOK
|
6.8 | IC50 | 3 | — | |
IEYYHWFOJFXPGP
|
6.8 | IC50 | 3 | — | |
BUDSAEMPVYFKML
|
6.8 | IC50 | 3 | — | |
PAISIGRMLVYIDB
|
6.8 | IC50 | 3 | — | |
GZADYKQLFNISTG
|
6.5 | IC50 | 2 | — | |
SAZVKYFGANAWRA
|
6.5 | IC50 | 3 | — | |
OMSYWTFGLFSMBY
|
6.4 | IC50 | 2 | — | |
CYJAZIKQEIQCOG
|
6.3 | IC50 | 2 | — | |
BEWRVZZHISITDQ
|
6.3 | IC50 | 3 | — | |
BEWRVZZHISITDQ
|
6.3 | IC50 | 3 | — | |
YSYQXQQIKOEBNN
|
6.3 | Ki | 3 | — | |
ZPHQKYQWQLYSDS
|
6.2 | IC50 | 3 | — | |
AATVMVZMTDKRJI
|
6.2 | IC50 | 3 | — | |
ZGOYLLCQBCBXHF
|
6.2 | IC50 | 3 | — | |
BUSBNAUESVLLQC
|
6.1 | IC50 | 3 | — | |
HNWIOZGMMTUVKP
|
6.0 | IC50 | 2 | — | |
NJCHEVDWMWFDNQ
|
6.0 | IC50 | 3 | — | |
MRXHFZNHXQEPNB
|
6.0 | Ki | 3 | — | |
PBYNWRKJSAGRFG
|
6.0 | IC50 | 2 | — |