Target Details
| UniProt AC | Q9NYY3 |
|---|---|
| Gene Symbol | PLK2 |
| Protein Name | Serine/threonine-protein kinase PLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 110
- Clinical molecules 10
- Avg pChEMBL 7.16
KEGG Pathways (1)
Active Molecules (110)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DZSUJUOJJJCWGG
|
7.2 | Ki | 55 | Yes | |
XFHCCTMTQFFLCT
|
7.1 | IC50 | 2 | — | |
JTYDPPQNZSHIQR
|
7.1 | IC50 | 2 | — | |
JETXRGKNZYUPEF
|
7.1 | IC50 | 6 | — | |
ITYGFIRONBGARW
|
7.1 | IC50 | 3 | — | |
FTVMYIRRFFYFIH
|
7.0 | IC50 | 3 | — | |
VINNOSMQDSWDTC
|
7.0 | IC50 | 3 | — | |
KPDOBADQSPMGFP
|
7.0 | IC50 | 3 | — | |
URBLFMVEDFWKGZ
|
7.0 | IC50 | 6 | — | |
AAWUJXDNCDOXTN
|
6.9 | IC50 | 3 | — | |
WPPGBVWZGMDXKF
|
6.9 | IC50 | 5 | — | |
MAULBJVKJOGNGD
|
6.9 | IC50 | 3 | — | |
BSFNGHCTZDCQBF
|
6.8 | Ki | 3 | — | |
JKZKKHVTLCFCGS
|
6.8 | IC50 | 3 | — | |
PVVRSMIEEGPASF
|
6.8 | IC50 | 3 | — | |
QMGCOLHGTKYVOP
|
6.8 | IC50 | 3 | — | |
KVJXBCZPOFTDAU
|
6.8 | IC50 | 2 | — | |
FMCBJKDUHHIOQB
|
6.7 | IC50 | 2 | — | |
HEVBIDCNQYUCRF
|
6.7 | IC50 | 2 | — | |
KHBSTEQSSXYFCY
|
6.7 | IC50 | 2 | — | |
PGHXJQMSVOKZRE
|
6.7 | IC50 | 3 | — | |
GCFCQBCBKXQUCD
|
6.7 | IC50 | 3 | — | |
ZDQJNYLFGPXANH
|
6.7 | IC50 | 3 | — | |
FVLMDPWEHBGZDD
|
6.6 | IC50 | 3 | — | |
WQQABBZFVHSXMU
|
6.6 | IC50 | 3 | — | |
LDFXILCAFQHTNH
|
6.6 | IC50 | 3 | — | |
NUQUWKXNHFMEAJ
|
6.6 | IC50 | 3 | — | |
MRITYVDXXFOOAU
|
6.6 | Kd | 6 | — | |
RNCCSJOQZGLCIQ
|
6.5 | IC50 | 3 | — | |
XDRHCUWKZRZSEP
|
6.5 | IC50 | 2 | — | |
KRFAHCVCYDZSOI
|
6.5 | IC50 | 2 | — | |
KSMYGTHXVJXRTI
|
6.5 | IC50 | 3 | — | |
AILANCLYZDKELS
|
6.5 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
6.5 | Kd | 289 | Yes | |
ZAJAQZFUONWQPQ
|
6.5 | IC50 | 3 | — | |
ZEHBZHZMQSHZFI
|
6.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.4 | IC50 | 408 | — | |
NERSFQYNEXMEPK
|
6.4 | IC50 | 3 | — | |
NCCZKHZUPCPIOT
|
6.4 | IC50 | 3 | — | |
KSNXWDGHPBZSBU
|
6.3 | IC50 | 2 | — | |
RJERVODZSCACGJ
|
6.3 | IC50 | 3 | — | |
ZHJGWYRLJUCMRT
|
6.3 | Kd | 18 | — | |
ANAAVHLLZPPWCU
|
6.3 | IC50 | 6 | — | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
SQRHNUCMJHZAKJ
|
6.2 | IC50 | 2 | — | |
CXPHUBRUHJPONW
|
6.2 | IC50 | 3 | — | |
NTVFVNYEAMJGDF
|
6.2 | IC50 | 3 | — | |
OSCRFGZIFNWYIZ
|
6.2 | IC50 | 3 | — | |
QIMUQYHRHHNTNY
|
6.2 | IC50 | 3 | — | |
AJJBWPRLFOMJCY
|
6.2 | IC50 | 3 | — |