Target Details
| UniProt AC | Q9NYY3 |
|---|---|
| Gene Symbol | PLK2 |
| Protein Name | Serine/threonine-protein kinase PLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 110
- Clinical molecules 10
- Avg pChEMBL 7.16
KEGG Pathways (1)
Active Molecules (110)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NDIUYMHNCUTVGE
|
8.7 | Ki | 25 | — | |
OXPLZKSKLWBEIM
|
8.7 | IC50 | 8 | Yes | |
PRMNYSLMFFRETJ
|
8.5 | IC50 | 3 | — | |
JSKUWFIZUALZLX
|
8.4 | Ki | 33 | — | |
DAAGOCSHXCDWDY
|
8.4 | IC50 | 3 | — | |
XANXBCMPWPUNSZ
|
8.4 | IC50 | 3 | — | |
OCYISXRMEJNANP
|
8.3 | IC50 | 3 | — | |
HKERRRNEVQHIRB
|
8.3 | IC50 | 2 | — | |
JMDRAMDTWLAOHD
|
8.3 | IC50 | 2 | — | |
SXNJFOWDRLKDSF
|
8.3 | IC50 | 3 | — | |
SXNJFOWDRLKDSF
|
8.3 | IC50 | 8 | — | |
CQQFCBITQKNHPX
|
8.2 | IC50 | 4 | — | |
XSTRJMHOLBBWNN
|
8.2 | IC50 | 4 | — | |
VMFNGGJHVCGNJO
|
8.2 | IC50 | 2 | — | |
JYYQJHRWOKIHGC
|
8.1 | IC50 | 3 | — | |
UEILKDPTXUZCFH
|
8.1 | IC50 | 3 | — | |
UMJFDLYATACWKW
|
8.1 | IC50 | 2 | — | |
GSXMJWLLQORXFR
|
8.1 | IC50 | 3 | — | |
TWYRQXNMQMYEGC
|
8.1 | IC50 | 2 | — | |
KOKNYBBQIVDZCK
|
8.1 | IC50 | 2 | — | |
UTHWBIPHRYUJSU
|
8.1 | IC50 | 11 | Yes | |
ZBJWJVGFIIULBV
|
8.0 | IC50 | 3 | — | |
QBQNTNGYPHAFJA
|
8.0 | IC50 | 2 | — | |
MOIBHLHUAXJLCW
|
7.9 | IC50 | 5 | — | |
DPROZSHCTFNYSW
|
7.9 | IC50 | 6 | Yes | |
QXAKKDDDYAESLJ
|
7.9 | IC50 | 6 | Yes | |
RHIJMDNVEPLDED
|
7.9 | IC50 | 2 | — | |
XQVVPGYIWAGRNI
|
7.9 | IC50 | 34 | — | |
UNZVQIJLQQYQLN
|
7.8 | IC50 | 6 | — | |
CIGSBKXHEYMHAF
|
7.8 | IC50 | 2 | — | |
NMVMZFAZMNUQMX
|
7.8 | IC50 | 2 | — | |
SFNMDOXBLCGZMQ
|
7.7 | IC50 | 3 | — | |
MCJYLZXJWVLMLI
|
7.7 | IC50 | 2 | — | |
XEXSGNRGTBSSOU
|
7.7 | IC50 | 3 | — | |
JPWPZFYYVIFSAZ
|
7.7 | IC50 | 3 | — | |
UMJFDLYATACWKW
|
7.7 | IC50 | 2 | — | |
UXNCNPVLRQGOMH
|
7.7 | IC50 | 3 | — | |
UZVJWQPORUUHRW
|
7.6 | IC50 | 3 | — | |
XEMJTISGDXHELX
|
7.6 | IC50 | 8 | Yes | |
GNFVJCMQLYMYRH
|
7.6 | IC50 | 2 | — | |
OYDGHJTZNAFKAQ
|
7.6 | IC50 | 6 | Yes | |
ZSYVDZWVCFZJLJ
|
7.5 | IC50 | 2 | — | |
OSCRFGZIFNWYIZ
|
7.5 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
VZDOSGQBGHVVCU
|
7.5 | IC50 | 3 | — | |
CAVRDKDHKZOOIF
|
7.4 | IC50 | 3 | — | |
NILXCNICWMPUMM
|
7.4 | IC50 | 2 | — | |
YOMURATVIWHSOR
|
7.3 | IC50 | 2 | — | |
PMMISILPBLQWSZ
|
7.2 | IC50 | 2 | — | |
MVYFNZROIDKPOZ
|
7.2 | IC50 | 3 | — |