Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VMHVFKJWJAKEES
|
6.7 | IC50 | 6 | — | |
VSVASKKCTHTYJG
|
6.7 | IC50 | 9 | — | |
VSVQHBIUNVDFOP
|
6.7 | IC50 | 6 | — | |
VYQTWOHAGUWLGB
|
6.7 | IC50 | 5 | — | |
VYQTWOHAGUWLGB
|
6.7 | IC50 | 5 | — | |
WAKCLPBZTLOHAP
|
6.7 | IC50 | 9 | — | |
WCUCMEYMHMWTGU
|
6.7 | IC50 | 6 | — | |
WDWVBDVZSOLQEF
|
6.7 | IC50 | 6 | — | |
WFSQFDUHZLJFOA
|
6.7 | IC50 | 6 | — | |
WKOBYQUPHFBDOX
|
6.7 | IC50 | 5 | — | |
WNTWPMDPWXFJJJ
|
6.7 | IC50 | 9 | — | |
WOSCFDBVQAKFEG
|
6.7 | IC50 | 5 | — | |
WTZPCQTWWNDNCQ
|
6.7 | IC50 | 6 | — | |
WVOMSZCXYDTSHK
|
6.7 | IC50 | 5 | — | |
XFHHYEOIODCSGJ
|
6.7 | IC50 | 6 | — | |
XFTSYFZIUPOJNI
|
6.7 | IC50 | 9 | — | |
XHVOFZVQIPBPRX
|
6.7 | IC50 | 6 | — | |
XMRPPWFWJKGYOU
|
6.7 | IC50 | 6 | — | |
XNMLEQBZPRKCFV
|
6.7 | IC50 | 5 | — | |
XODVORNLEGKQIG
|
6.7 | IC50 | 2 | — | |
XQLZXHQTAMMUIE
|
6.7 | IC50 | 6 | — | |
XWKQZYOSWGEGIH
|
6.7 | IC50 | 7 | — | |
XWOQCKJZIGPMAB
|
6.7 | IC50 | 9 | — | |
XZXJVMPFESCWIA
|
6.7 | IC50 | 6 | — | |
XZXJVMPFESCWIA
|
6.7 | IC50 | 6 | — | |
YBWWKUHCOLJULU
|
6.7 | IC50 | 6 | — | |
YGVSSBPHNLLAHU
|
6.7 | IC50 | 9 | — | |
YOKJZKNQSMSTEA
|
6.7 | IC50 | 6 | — | |
YTRWVNINOQGWBU
|
6.7 | IC50 | 9 | — | |
ZFCGKKJTVIQDQQ
|
6.7 | IC50 | 6 | — | |
ZNXLTLNJAJGULG
|
6.7 | IC50 | 4 | — | |
ZQTYCYKZVIURPR
|
6.7 | IC50 | 6 | — | |
ZRYDQZBXQILIHI
|
6.7 | IC50 | 5 | — | |
ZSFSNNXZQSIUQS
|
6.7 | IC50 | 5 | — | |
ZSXNAVZVCNPEOT
|
6.7 | IC50 | 6 | — | |
ZVQWWSRTRLSWBL
|
6.7 | IC50 | 6 | — | |
ZWXSRTQVEQAVMT
|
6.7 | IC50 | 7 | — | |
ZYKQSVFRGAYPFG
|
6.7 | IC50 | 5 | — | |
ZYRQHVIUTUPUQS
|
6.7 | IC50 | 9 | — | |
AWAHFDYWQKGERT
|
6.7 | IC50 | 2 | — | |
SLIFZZITPODXKX
|
6.7 | IC50 | 6 | — | |
KAERLKBLDZCEHI
|
6.7 | IC50 | 2 | — | |
LTHGSGNCNMDKSD
|
6.7 | IC50 | 9 | — | |
HMZGUBXDLSCJRA
|
6.6 | IC50 | 2 | — | |
AXERCKVGIICWDT
|
6.6 | IC50 | 7 | — | |
BGFSBIGNWZKZAG
|
6.6 | IC50 | 2 | — | |
CIECLIQCGMZLNI
|
6.6 | IC50 | 7 | — | |
CKXQPVNWDKKSSJ
|
6.6 | IC50 | 7 | — | |
CMILELPCKPBWNV
|
6.6 | IC50 | 4 | — | |
CYWJCWFAPFOQOP
|
6.6 | IC50 | 7 | — |