Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OWSWNWFBDKDKGQ
|
6.7 | IC50 | 6 | — | |
PAQBVDRSJSOVGY
|
6.7 | IC50 | 9 | — | |
PCDLASLXDUVOPP
|
6.7 | IC50 | 6 | — | |
PDCIXCSHUGGJPD
|
6.7 | IC50 | 9 | — | |
PGVLOHBGJFPPRB
|
6.7 | IC50 | 9 | — | |
PLPINOJFYBYYDH
|
6.7 | IC50 | 6 | — | |
PNLMCNAXDCPSHW
|
6.7 | IC50 | 5 | — | |
PNLMCNAXDCPSHW
|
6.7 | IC50 | 6 | — | |
PSUOIOJISBKJMX
|
6.7 | IC50 | 6 | — | |
PTUHEHLILKOCKH
|
6.7 | IC50 | 9 | — | |
PUPUVPPZPABPSG
|
6.7 | IC50 | 6 | — | |
QAJSSTGAGZUFTN
|
6.7 | IC50 | 7 | — | |
QIPWIFGPTSTIPS
|
6.7 | IC50 | 6 | — | |
QOFPGIURZHAJIH
|
6.7 | IC50 | 6 | — | |
QWTLJZSIFBCFBX
|
6.7 | IC50 | 7 | — | |
QWTLJZSIFBCFBX
|
6.7 | IC50 | 6 | — | |
QYHLJTSUFLTMRN
|
6.7 | IC50 | 9 | — | |
RAPGDNCSRYGONO
|
6.7 | IC50 | 6 | — | |
RMQZFHNZKHTFFQ
|
6.7 | IC50 | 6 | — | |
RNEYCMVMZFAUCY
|
6.7 | IC50 | 6 | — | |
RPWBQONKJLUMGK
|
6.7 | IC50 | 6 | — | |
RQJCTXCBKQJXOV
|
6.7 | IC50 | 5 | — | |
RUDYLSGWPPPMGZ
|
6.7 | IC50 | 6 | — | |
RVWHBLSSCKUHRD
|
6.7 | IC50 | 7 | — | |
RYCWVDJHDBTEEA
|
6.7 | IC50 | 6 | — | |
RZDDODLDFHUUSO
|
6.7 | IC50 | 9 | — | |
SCJNYBYSTCRPAO
|
6.7 | IC50 | 7 | — | |
SELGYLPDJDLPJJ
|
6.7 | IC50 | 5 | — | |
SHUANTOYSJCYHF
|
6.7 | IC50 | 7 | — | |
SIKSLMHBJBRHAP
|
6.7 | IC50 | 6 | — | |
SOEGPCFMFUKWHZ
|
6.7 | IC50 | 6 | — | |
SPKNPIWZWPDFPY
|
6.7 | IC50 | 6 | — | |
SPLVLYILTZEOKC
|
6.7 | IC50 | 9 | — | |
SQIRDMQXJCPDHP
|
6.7 | IC50 | 6 | — | |
SRSLIRBECCWKOE
|
6.7 | IC50 | 6 | — | |
SUQQDRCRQDKHCI
|
6.7 | IC50 | 9 | — | |
SUQQDRCRQDKHCI
|
6.7 | IC50 | 6 | — | |
SZFFNMGIXIMKFV
|
6.7 | IC50 | 6 | — | |
TXZFORDUGWJTSQ
|
6.7 | IC50 | 9 | — | |
TZAZCOVOUHIOIH
|
6.7 | IC50 | 9 | — | |
UFRQWZYUZLYCRM
|
6.7 | IC50 | 5 | — | |
UKTQALXBQGWLKL
|
6.7 | IC50 | 6 | — | |
UODNLJWDEILUIA
|
6.7 | IC50 | 6 | — | |
UTRWOQWGKFKJDY
|
6.7 | IC50 | 6 | — | |
UTWMDDZNYDDKPY
|
6.7 | IC50 | 6 | — | |
UULJMLAHWBWQBO
|
6.7 | IC50 | 6 | — | |
UWGQTQNIPQDTSH
|
6.7 | IC50 | 9 | — | |
UWGQTQNIPQDTSH
|
6.7 | IC50 | 9 | — | |
VBXUAFKZCVKOQN
|
6.7 | IC50 | 5 | — | |
VLRNVSCGMBELQB
|
6.7 | IC50 | 6 | — |