Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HEZCSXMOOAADBW
|
6.7 | IC50 | 6 | — | |
HKSXMVBEMPZHJC
|
6.7 | IC50 | 7 | — | |
HOWNBGZWAXBZST
|
6.7 | IC50 | 6 | — | |
HTNQYVUPMKKVPR
|
6.7 | IC50 | 6 | — | |
IIPGUOQKZWUTQB
|
6.7 | IC50 | 6 | — | |
IJMXMWWSKLBXFF
|
6.7 | IC50 | 5 | — | |
IJQBKJGUIDXXLI
|
6.7 | IC50 | 9 | — | |
IJQBKJGUIDXXLI
|
6.7 | IC50 | 5 | — | |
ISQDCYJPZNRXLS
|
6.7 | IC50 | 2 | — | |
IZDUIVZZOXJQKT
|
6.7 | IC50 | 9 | — | |
IZRVAAWMOPBZGL
|
6.7 | IC50 | 5 | — | |
JASLFJDPMFIVTK
|
6.7 | IC50 | 5 | — | |
JCEFHFGLYRFDSK
|
6.7 | IC50 | 5 | — | |
JEFBXCSJCMHIIO
|
6.7 | IC50 | 7 | — | |
JFCFXMMAWHGRMB
|
6.7 | IC50 | 7 | — | |
JHMADRGGYHZRPX
|
6.7 | IC50 | 5 | — | |
JMDJVTKHPSFJBK
|
6.7 | IC50 | 6 | — | |
JPRFEVKWGIBMIH
|
6.7 | IC50 | 6 | — | |
JPSORPODXWGJEF
|
6.7 | IC50 | 5 | — | |
JYGHIHQUUSIMSX
|
6.7 | IC50 | 6 | — | |
KEIIBASGNFWEPN
|
6.7 | IC50 | 2 | — | |
KJJMNWWMDYYZSU
|
6.7 | IC50 | 2 | — | |
KJXFLZZKFSETJZ
|
6.7 | IC50 | 5 | — | |
KLDQRWLIWJOZMA
|
6.7 | IC50 | 6 | — | |
KLLLDNLYQNAKOW
|
6.7 | IC50 | 6 | — | |
KNKBXFUDTNASDX
|
6.7 | IC50 | 6 | — | |
KNOSKPVYWKOAAP
|
6.7 | IC50 | 5 | — | |
KWUIXBNQNOVRJJ
|
6.7 | IC50 | 6 | — | |
LAABYGDZDAENTA
|
6.7 | IC50 | 6 | — | |
LBVWNRFNOZHXGU
|
6.7 | IC50 | 6 | — | |
LOVXTLJVBKIDNT
|
6.7 | IC50 | 9 | — | |
LTNGKOAIMLLMQU
|
6.7 | IC50 | 9 | — | |
LWTPFXMUZKOEMR
|
6.7 | IC50 | 5 | — | |
MBUFHYIDRFQNFX
|
6.7 | IC50 | 6 | — | |
MJLQPTUXPJMBNG
|
6.7 | IC50 | 9 | — | |
MMORELYIVNMTSR
|
6.7 | IC50 | 5 | — | |
MTLJCKRPLWHNCD
|
6.7 | IC50 | 2 | — | |
MVGDWWDXFJNLNG
|
6.7 | IC50 | 9 | — | |
NEFGSTFCOAETMW
|
6.7 | IC50 | 6 | — | |
NFIYWRAMGWCCKU
|
6.7 | IC50 | 6 | — | |
NHIOUCSDAKKLBQ
|
6.7 | IC50 | 7 | — | |
NIIPWXCPEONJIK
|
6.7 | IC50 | 6 | — | |
NKZTUIQTQVDTRI
|
6.7 | IC50 | 5 | — | |
NOHFWDPNSURDSS
|
6.7 | IC50 | 7 | — | |
NRIQXUKIFJKSBE
|
6.7 | IC50 | 5 | — | |
NSUOMXJJQZTYBL
|
6.7 | IC50 | 6 | — | |
NWLLJGVSVSXYSN
|
6.7 | IC50 | 5 | — | |
OJCCNWLOIVOTIV
|
6.7 | IC50 | 2 | — | |
OLNGHVOKJOVKDT
|
6.7 | IC50 | 5 | — | |
OOOSVTAESCWYNL
|
6.7 | IC50 | 6 | — |