Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNUOLEFJKLTZAN
|
7.0 | IC50 | 2 | — | |
XRPROGLAYMHNAO
|
7.0 | IC50 | 2 | — | |
YUQHSQMKLJXSFR
|
7.0 | IC50 | 2 | — | |
ZDUPHHYECRNJFI
|
7.0 | IC50 | 2 | — | |
ZGNYHIFMOOIDJG
|
7.0 | IC50 | 2 | — | |
DIIRGFRZMVBYSW
|
7.0 | IC50 | 8 | — | |
HVFVQLFPRQYJTR
|
7.0 | IC50 | 2 | — | |
VVLLRESVVUQNTP
|
7.0 | IC50 | 2 | — | |
VBWQPLLCGUWXEE
|
7.0 | IC50 | 5 | — | |
VJFZHLXFXHOTLG
|
7.0 | IC50 | 4 | — | |
JEWRIBSMLSEECE
|
7.0 | IC50 | 8 | — | |
QAMWYSGCQVRMCX
|
6.9 | IC50 | 2 | — | |
CSFFNUBEOYPGPP
|
6.9 | IC50 | 2 | — | |
DKHFQORSZZALIY
|
6.9 | IC50 | 2 | — | |
VFRSDNYJPASDOG
|
6.9 | IC50 | 2 | — | |
YUBVKTOENBVBLZ
|
6.9 | IC50 | 2 | — | |
SVNPEEHTDUPXBZ
|
6.9 | IC50 | 2 | — | |
JNKXYDCPHHUMKG
|
6.9 | IC50 | 4 | — | |
JNKXYDCPHHUMKG
|
6.9 | IC50 | 2 | — | |
LWOAAFPWDPZGMV
|
6.9 | IC50 | 2 | — | |
HZZNUWNFLHMBRW
|
6.9 | IC50 | 9 | — | |
OUDPXOAJUACLFI
|
6.9 | IC50 | 2 | — | |
KKBGPXKESUWDQK
|
6.8 | IC50 | 2 | — | |
DSXXEELGXBCYNQ
|
6.8 | IC50 | 28 | Yes | |
UNLGDKYAZYKOQD
|
6.8 | IC50 | 2 | — | |
OSIQEILYTOCUHB
|
6.8 | IC50 | 2 | — | |
VSBGARFTIZDELR
|
6.8 | IC50 | 2 | — | |
DMUSMYYDKCXFKR
|
6.8 | IC50 | 8 | — | |
DQFXKZPDQHUJLY
|
6.8 | IC50 | 8 | — | |
RXVKNJWYFKQBNZ
|
6.8 | IC50 | 2 | — | |
UCRLRCYXXQTIRC
|
6.8 | IC50 | 7 | — | |
WXFNPYZGKHGERJ
|
6.8 | IC50 | 7 | — | |
BIIVYFLTOXDAOV
|
6.8 | Kd | 82 | Yes | |
JDTTVEQCHMEDBM
|
6.8 | IC50 | 2 | — | |
LKIOJDJYOLZKMP
|
6.8 | IC50 | 2 | — | |
MHGIJKPXAGPHGD
|
6.8 | IC50 | 2 | — | |
RUBYHLPRZRMTJO
|
6.8 | IC50 | 3 | — | |
RUBYHLPRZRMTJO
|
6.8 | IC50 | 7 | — | |
RUBYHLPRZRMTJO
|
6.8 | IC50 | 3 | — | |
VJFWDARVZBIZDG
|
6.8 | IC50 | 2 | — | |
NUZCHSPIOISCKD
|
6.8 | IC50 | 2 | — | |
FECJFYFWBIAIIL
|
6.8 | IC50 | 4 | — | |
OUSFTKFNBAZUKL
|
6.8 | Kd | 58 | Yes | |
DWPSXXHIBIAPLR
|
6.8 | IC50 | 2 | — | |
NJVMZQYUJOCBPO
|
6.8 | IC50 | 2 | — | |
DMUSMYYDKCXFKR
|
6.7 | IC50 | 9 | — | |
VXLAKHWYGRKCGI
|
6.7 | IC50 | 9 | — | |
WIJLQVQUQLNZFD
|
6.7 | IC50 | 2 | — | |
GOOZCRGJKQVEFX
|
6.7 | IC50 | 2 | — | |
CIRXEIZEFCEWTH
|
6.7 | IC50 | 2 | — |