Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DBHDGUFCNJWVQW
|
7.0 | IC50 | 2 | — | |
YDHKLKQGRRFWHD
|
7.0 | IC50 | 8 | — | |
FSELUFUYNUNZKD
|
7.0 | Kd | 4 | — | |
AFGVRZRGTJRSPW
|
7.0 | IC50 | 2 | — | |
BCDWZDLKBNFZAG
|
7.0 | IC50 | 2 | — | |
BCDWZDLKBNFZAG
|
7.0 | IC50 | 2 | — | |
BRVCJFXSVHNURA
|
7.0 | IC50 | 2 | — | |
CIPOPUVTFAXGFK
|
7.0 | IC50 | 2 | — | |
CLKHZAFUFOHOBR
|
7.0 | IC50 | 2 | — | |
CMRKMABDVBMJKO
|
7.0 | IC50 | 2 | — | |
CVLHTCTYABLZJG
|
7.0 | IC50 | 2 | — | |
CWHZJISLECRIEV
|
7.0 | IC50 | 2 | — | |
GBFWJIWBIXTABL
|
7.0 | IC50 | 2 | — | |
GDQXJQSQYMMKRA
|
7.0 | IC50 | 15 | — | |
GFGVTCZTOKDNKE
|
7.0 | IC50 | 2 | — | |
GLRFVOOMFBLXQE
|
7.0 | IC50 | 2 | — | |
HIKHKAPMLNZMCE
|
7.0 | IC50 | 2 | — | |
HSKSOLAQHJHQHZ
|
7.0 | IC50 | 2 | — | |
HSUGNMZPSHOTNZ
|
7.0 | IC50 | 2 | — | |
INBVJLOENDWCKQ
|
7.0 | IC50 | 2 | — | |
IOKMWEQZOAUPMW
|
7.0 | IC50 | 2 | — | |
IRMKVBJNYMQMDC
|
7.0 | IC50 | 2 | — | |
JAJQGAQWIYQLJV
|
7.0 | IC50 | 2 | — | |
JJGMBFIFSOWZTR
|
7.0 | IC50 | 2 | — | |
JLZQRZCGFZRBJQ
|
7.0 | IC50 | 2 | — | |
KWESRLQUCSBVEY
|
7.0 | IC50 | 2 | — | |
LXGBKZHEQNMKJY
|
7.0 | IC50 | 2 | — | |
MBFKYSMHWKYPEB
|
7.0 | IC50 | 2 | — | |
MFOJDWXAHANYHN
|
7.0 | IC50 | 2 | — | |
MGUQQNVMCQNVCL
|
7.0 | IC50 | 2 | — | |
MQKFDLRVYBCIPL
|
7.0 | IC50 | 2 | — | |
MYVBEOAIEAODMH
|
7.0 | IC50 | 2 | — | |
MZLQTHFOMLFMOR
|
7.0 | IC50 | 2 | — | |
NESVUGQFAJABNV
|
7.0 | IC50 | 2 | — | |
NIDWYRMRHGIQIV
|
7.0 | IC50 | 2 | — | |
NSMMAQNNMFYEHG
|
7.0 | IC50 | 2 | — | |
PAPOIMUQKDYWOG
|
7.0 | IC50 | 2 | — | |
PNSNIUNNSOVHCB
|
7.0 | IC50 | 2 | — | |
PRGGODNOOBWDLY
|
7.0 | IC50 | 2 | — | |
QFPDYVCUELOMKG
|
7.0 | IC50 | 2 | — | |
QFPDYVCUELOMKG
|
7.0 | IC50 | 2 | — | |
QVWJCPCDKVFGTB
|
7.0 | IC50 | 7 | — | |
RIJUYHRORZYQRY
|
7.0 | IC50 | 2 | — | |
RRVNPAIZDWDNFC
|
7.0 | IC50 | 2 | — | |
RSKFCQGPFNRQIQ
|
7.0 | IC50 | 2 | — | |
SYARFBBVLGMUMN
|
7.0 | IC50 | 2 | — | |
VHMWWZAIMFNMRD
|
7.0 | IC50 | 2 | — | |
VTABUZXCILJXEW
|
7.0 | IC50 | 2 | — | |
VVJGKNRGWCNPOY
|
7.0 | IC50 | 2 | — | |
WLDONHMIFMWHAZ
|
7.0 | IC50 | 2 | — |