Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MJOVPABKFQFAHK
|
6.0 | IC50 | 7 | — | |
MPOVNMQJTKXOAG
|
6.0 | IC50 | 2 | — | |
MUVWORKUAAGULV
|
6.0 | IC50 | 2 | — | |
NIDDSEZQRJOBEU
|
6.0 | IC50 | 2 | — | |
NLFIKRGSUXUBRO
|
6.0 | IC50 | 2 | — | |
NNNLDSYGAMOLGZ
|
6.0 | IC50 | 2 | — | |
NWAPJLWXJZKRKW
|
6.0 | IC50 | 2 | — | |
OCDGUPGJTXDKQV
|
6.0 | IC50 | 2 | — | |
OOOTWPYQOQWVHB
|
6.0 | IC50 | 2 | — | |
OPOLXEPGMNZIEN
|
6.0 | IC50 | 4 | — | |
QGCDJVRAMTZHTL
|
6.0 | IC50 | 2 | — | |
QMKWCYQYIVXOCQ
|
6.0 | IC50 | 2 | — | |
RIPKUAOEAZQYSR
|
6.0 | IC50 | 2 | — | |
RIPKUAOEAZQYSR
|
6.0 | IC50 | 2 | — | |
RVJPXDTZPIJZCS
|
6.0 | IC50 | 2 | — | |
SBDXQNJXPIKHRC
|
6.0 | IC50 | 2 | — | |
SIGKFKBFXQQJJH
|
6.0 | IC50 | 7 | — | |
SJOAZCQZGBQZMY
|
6.0 | IC50 | 2 | — | |
SKWBROMFZCGGTH
|
6.0 | IC50 | 2 | — | |
SLLQPTPVVMWBIH
|
6.0 | IC50 | 2 | — | |
UAEGJOAMXWXUPW
|
6.0 | IC50 | 2 | — | |
UHNVQQQSPQBPSF
|
6.0 | IC50 | 2 | — | |
UQDLBEGORWSOQS
|
6.0 | IC50 | 7 | — | |
UQJPTNCNWZZWPZ
|
6.0 | IC50 | 2 | — | |
VCKVKJIEERRCGQ
|
6.0 | IC50 | 2 | — | |
VITZAEMGPINHJI
|
6.0 | IC50 | 2 | — | |
VMOGYLIDBJZEGI
|
6.0 | IC50 | 2 | — | |
XGHGKGOFDKUMIW
|
6.0 | IC50 | 2 | — | |
XIQDZYPJMAGASL
|
6.0 | IC50 | 2 | — | |
XOSLXBCBLVUKRT
|
6.0 | IC50 | 2 | — | |
YEUXYLMZOGKIDT
|
6.0 | IC50 | 2 | — | |
YGZVFEAVMKDQGV
|
6.0 | IC50 | 2 | — | |
YXOUVVXABJCBBF
|
6.0 | IC50 | 2 | — | |
ZDHKGXKBNMHPPE
|
6.0 | IC50 | 2 | — | |
ZLPCBGQKMZEQMX
|
6.0 | IC50 | 2 | — | |
ZPFYVLDGCDZJCW
|
6.0 | IC50 | 2 | — | |
ZSZQVQMTHDDMRZ
|
6.0 | IC50 | 2 | — |