Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AMJAYGUNGYXSFK
|
6.0 | IC50 | 2 | — | |
BEQMGVFFCIVCEU
|
6.0 | IC50 | 2 | — | |
BHDLEDZNDSWKRP
|
6.0 | IC50 | 2 | — | |
BJJLPBXVKCFYLZ
|
6.0 | IC50 | 2 | — | |
BJQKZYVLMUWQLN
|
6.0 | IC50 | 2 | — | |
BMFJNINKASGUDG
|
6.0 | IC50 | 2 | — | |
BQDIUOURYAGTEW
|
6.0 | IC50 | 2 | — | |
BQOGUYSNUZLDDP
|
6.0 | IC50 | 2 | — | |
BWDKJJRENSRLOR
|
6.0 | IC50 | 2 | — | |
BXOKOMSBDLPWMM
|
6.0 | IC50 | 2 | — | |
CCGMCVDHWFZTLR
|
6.0 | IC50 | 2 | — | |
CCGMCVDHWFZTLR
|
6.0 | IC50 | 2 | — | |
CEQCQJCJVFCCHG
|
6.0 | IC50 | 2 | — | |
CQQXEFOKQUOYBV
|
6.0 | IC50 | 2 | — | |
CTFVTQDBNNPXAX
|
6.0 | IC50 | 7 | — | |
DFOCZNXPBFUNKX
|
6.0 | IC50 | 2 | — | |
DKYHVNFDJFQDLQ
|
6.0 | IC50 | 2 | — | |
DOTQQXIKDOWYKJ
|
6.0 | IC50 | 2 | — | |
DPMXWSJCLPNLDJ
|
6.0 | IC50 | 2 | — | |
DQFFHODWODODSN
|
6.0 | IC50 | 2 | — | |
DRGGVGJKEXYMTJ
|
6.0 | IC50 | 2 | — | |
DWWSHEDDRAZIRR
|
6.0 | IC50 | 2 | — | |
FCEDZVAVRKXWMU
|
6.0 | IC50 | 2 | — | |
FCEDZVAVRKXWMU
|
6.0 | IC50 | 2 | — | |
FCIPPCSOLCGGSL
|
6.0 | IC50 | 2 | — | |
FCIPPCSOLCGGSL
|
6.0 | IC50 | 2 | — | |
GBFWJIWBIXTABL
|
6.0 | IC50 | 2 | — | |
GBJZOTFIIJHFPO
|
6.0 | IC50 | 2 | — | |
GFWXCQGWQBHGSR
|
6.0 | IC50 | 2 | — | |
GNWKOJILXOCBIH
|
6.0 | IC50 | 2 | — | |
GRBMJJYBCNETMC
|
6.0 | IC50 | 2 | — | |
GWRDYNFOVJSTIH
|
6.0 | IC50 | 2 | — | |
HQFIWJKVWLGQPU
|
6.0 | IC50 | 2 | — | |
HZOOEMDJXGKULR
|
6.0 | IC50 | 2 | — | |
HZOOEMDJXGKULR
|
6.0 | IC50 | 2 | — | |
IGYWYLYPEQDROD
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JAJQGAQWIYQLJV
|
6.0 | IC50 | 2 | — | |
JOWUQFXKZMRBLF
|
6.0 | IC50 | 2 | — | |
KFZHSFKSGFAJRH
|
6.0 | IC50 | 2 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KVXQLXPFDZNTJA
|
6.0 | IC50 | 2 | — | |
LBCMJGKNZDHRGC
|
6.0 | IC50 | 2 | — | |
LDWCNQNKYXQESA
|
6.0 | IC50 | 2 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MAIUJHAMFJOCMD
|
6.0 | IC50 | 2 | — | |
MBCSGTXFDOYTJD
|
6.0 | IC50 | 2 | — | |
MBEIKTZUWOZUCQ
|
6.0 | IC50 | 2 | — | |
MGVAVLHGVGIHBX
|
6.0 | IC50 | 2 | — | |
MJIAIWZDAWCWQS
|
6.0 | IC50 | 2 | — |