Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NZPIEKMSIASRGO
|
6.3 | IC50 | 2 | — | |
NZPOEPQZJYEBFF
|
6.3 | IC50 | 2 | — | |
ODVHBZWGFUQUGC
|
6.3 | IC50 | 2 | — | |
OGTBLGPHNBOWNQ
|
6.3 | IC50 | 2 | — | |
OSRZLJBASCMYIV
|
6.3 | IC50 | 2 | — | |
PNGJRQBFSPHWPR
|
6.3 | IC50 | 2 | — | |
PVKHAVSZQDRVDJ
|
6.3 | IC50 | 2 | — | |
QCSAEDFGKQLNLB
|
6.3 | IC50 | 2 | — | |
QKALFVARZSPOPP
|
6.3 | IC50 | 2 | — | |
QNOLRWWPCXIDMS
|
6.3 | IC50 | 2 | — | |
QUKRFGLEZVLWKV
|
6.3 | IC50 | 2 | — | |
REPHJBKSOJHVNS
|
6.3 | IC50 | 2 | — | |
REPHJBKSOJHVNS
|
6.3 | IC50 | 2 | — | |
RHCRAQAIFNGFBJ
|
6.3 | IC50 | 2 | — | |
RSMDTXWYRFXKRV
|
6.3 | IC50 | 2 | — | |
SRZPRAQMUBZZJC
|
6.3 | IC50 | 2 | — | |
SSSTXJLNCJNBQR
|
6.3 | IC50 | 2 | — | |
UNOKYGYYXZESEA
|
6.3 | IC50 | 2 | — | |
URJZAWIKZMCHJX
|
6.3 | IC50 | 2 | — | |
UZTJYPIRNJRKRO
|
6.3 | IC50 | 2 | — | |
VVVYIXNVAPSYSE
|
6.3 | IC50 | 3 | — | |
VWEAURJRFYXAIC
|
6.3 | IC50 | 2 | — | |
VXHBMDURWBXUCT
|
6.3 | IC50 | 2 | — | |
XGHIYHCQTGULDC
|
6.3 | IC50 | 2 | — | |
XGHIYHCQTGULDC
|
6.3 | IC50 | 2 | — | |
XPQIZMPKQACYQI
|
6.3 | IC50 | 2 | — | |
XWDLESVCEJCONG
|
6.3 | IC50 | 2 | — | |
YDQNOXVOVMJWBB
|
6.3 | IC50 | 2 | — | |
YGPHRCFUAUVVJJ
|
6.3 | IC50 | 2 | — | |
YLWJFVVLDWOHSZ
|
6.3 | IC50 | 2 | — | |
YSXLTPKOHLVCRQ
|
6.3 | IC50 | 2 | — | |
ZLWRADBWHLXEKI
|
6.3 | IC50 | 2 | — | |
VYKCLMALANGCDF
|
6.2 | IC50 | 6 | — | |
KUPBLGREELQEBD
|
6.2 | IC50 | 2 | — | |
URLDJGLPRNVRMR
|
6.2 | IC50 | 2 | — | |
XZMGOWQHLJWQJN
|
6.2 | IC50 | 2 | — | |
ZDEBEWQYXJZQRS
|
6.2 | IC50 | 12 | — | |
FWLMVFUGMHIOAA
|
6.1 | Kd | 26 | — | |
OETLNMOJNONWOY
|
6.1 | IC50 | 4 | — | |
OUDPXOAJUACLFI
|
6.1 | IC50 | 2 | — | |
WCEHIDWONYOKOJ
|
6.1 | IC50 | 2 | — | |
HJNYNZZNOGDODX
|
6.1 | IC50 | 7 | — | |
BECZMWHGUIMQOD
|
6.1 | IC50 | 8 | — | |
GGKAQFSAJDFYOL
|
6.0 | IC50 | 3 | — | |
JHQMFXCXGIEJNS
|
6.0 | IC50 | 2 | — | |
NFYBILFYIVKJHJ
|
6.0 | IC50 | 2 | — | |
OBJNFLYHUXWUPF
|
6.0 | IC50 | 17 | — | |
ZQLILUVVXPRXLE
|
6.0 | IC50 | 3 | — | |
XLSYZSRXVVCHLS
|
6.0 | Kd | 48 | — | |
ABBONWAQWSLIBJ
|
6.0 | IC50 | 2 | — |