Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WFWFIAFTMSUDNO
|
6.4 | IC50 | 7 | — | |
BPWZJVKIVHVVHP
|
6.4 | IC50 | 2 | — | |
OOYJNUNOVRCHJZ
|
6.4 | IC50 | 2 | — | |
VFWVTIHYVUKNGR
|
6.4 | IC50 | 2 | — | |
SIUIDAWJHAGUSX
|
6.4 | IC50 | 2 | — | |
YZCUMZWULWOUMD
|
6.4 | IC50 | 4 | — | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
IXAUUWHGCOSTKM
|
6.3 | IC50 | 2 | — | |
OMLLDMWWOBOZOL
|
6.3 | IC50 | 2 | — | |
GESCLFJYHIIAJV
|
6.3 | IC50 | 2 | — | |
ANAUELZVFNQHDD
|
6.3 | IC50 | 2 | — | |
ANAUELZVFNQHDD
|
6.3 | IC50 | 2 | — | |
ANQSXTYKVYGWEU
|
6.3 | IC50 | 2 | — | |
BEJOEUYZEIRAQE
|
6.3 | IC50 | 2 | — | |
BWHBJRMIXAHYNP
|
6.3 | IC50 | 2 | — | |
BXLFDQKBLYJUDW
|
6.3 | IC50 | 2 | — | |
CFSQJURXJXPCHZ
|
6.3 | IC50 | 2 | — | |
CLZRKIMYXQSYDV
|
6.3 | IC50 | 2 | — | |
CQEDXPZMGJKPPO
|
6.3 | IC50 | 2 | — | |
DFIYSRMKKAAUCG
|
6.3 | IC50 | 2 | — | |
FCVZMQKLBJRTIJ
|
6.3 | IC50 | 2 | — | |
FEGMAABADHKFRL
|
6.3 | IC50 | 2 | — | |
FMOQVRHJLGKPQM
|
6.3 | IC50 | 2 | — | |
GBRRMEYNRGRWIF
|
6.3 | IC50 | 2 | — | |
GYGOEUUUEBBBSA
|
6.3 | IC50 | 2 | — | |
HAPMPJQMNDISFK
|
6.3 | IC50 | 2 | — | |
HFHCVACHWOBZSK
|
6.3 | IC50 | 2 | — | |
HFXBWCYAICXNTK
|
6.3 | IC50 | 2 | — | |
ICJODIJVTMFAFW
|
6.3 | IC50 | 2 | — | |
IMZPHTNNVQUJCC
|
6.3 | IC50 | 2 | — | |
IPKOJRIIIDKFPB
|
6.3 | IC50 | 2 | — | |
ISIYHJMGMMBACO
|
6.3 | IC50 | 2 | — | |
JFSZDNXDUFONBS
|
6.3 | IC50 | 2 | — | |
JRHODUWDJJDIBX
|
6.3 | IC50 | 2 | — | |
JWMVMNLDZDYLCQ
|
6.3 | IC50 | 2 | — | |
KAVMCMWWFGWRQL
|
6.3 | IC50 | 2 | — | |
KMMBIJYVDWRKBD
|
6.3 | IC50 | 2 | — | |
LKUYDGNZVRTSGY
|
6.3 | IC50 | 2 | — | |
LMESFSCXDXXDRB
|
6.3 | IC50 | 2 | — | |
LMXJFHNFBODOER
|
6.3 | IC50 | 2 | — | |
LOIKMRHDZMIQPQ
|
6.3 | IC50 | 2 | — | |
LOSJMKRETYYECE
|
6.3 | IC50 | 2 | — | |
LSVXYJZKVKXKPP
|
6.3 | IC50 | 2 | — | |
MATPVGHWQGMDHM
|
6.3 | IC50 | 2 | — | |
MAVBTVKDGBLESI
|
6.3 | IC50 | 2 | — | |
MVPNCGHIJZPZTK
|
6.3 | IC50 | 2 | — | |
NFZCREOZCARLGQ
|
6.3 | IC50 | 2 | — | |
NKCQMMBCQQEIBL
|
6.3 | IC50 | 2 | — | |
NPPHHOUDISHMQN
|
6.3 | IC50 | 2 | — | |
NRZCIWFWFPDAAI
|
6.3 | IC50 | 2 | — |