Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DKIOTQWXLYOBOF
|
6.6 | IC50 | 7 | — | |
DKNAZEYWKWYKJO
|
6.6 | IC50 | 7 | — | |
DLVVFKMWFVZWDD
|
6.6 | IC50 | 7 | — | |
FALPBHNCTNGUFH
|
6.6 | IC50 | 7 | — | |
FSJGFYIBZOXTAU
|
6.6 | IC50 | 7 | — | |
GQFCNTKPAFRBKK
|
6.6 | IC50 | 5 | — | |
HRHHBYMFSQGBEX
|
6.6 | IC50 | 7 | — | |
HUKPFWLRPMADDJ
|
6.6 | IC50 | 7 | — | |
HWTFMLLJQLAKMY
|
6.6 | IC50 | 7 | — | |
IEVJHGZSBPGTMO
|
6.6 | IC50 | 3 | — | |
IHOAWPUMJLGVEZ
|
6.6 | IC50 | 7 | — | |
ILLVNLODYLPPIC
|
6.6 | IC50 | 7 | — | |
IOZSUUYSURMXEI
|
6.6 | IC50 | 7 | — | |
IUJVWZRIKASHNS
|
6.6 | IC50 | 7 | — | |
IXRHEVMMVUNFRH
|
6.6 | IC50 | 7 | — | |
JKHQLEAMZNVIPI
|
6.6 | IC50 | 7 | — | |
JMVIDMZVTXZHKA
|
6.6 | IC50 | 7 | — | |
LNYCRXZEMSCWFG
|
6.6 | IC50 | 7 | — | |
LRKRQTMUHJKJQW
|
6.6 | IC50 | 7 | — | |
NLZHDSMHJXZJTG
|
6.6 | IC50 | 7 | — | |
OBHIERMOPIJJOL
|
6.6 | IC50 | 4 | — | |
PWIPCKSOLCEBRW
|
6.6 | IC50 | 2 | — | |
QSERWBXLEKAYCJ
|
6.6 | IC50 | 7 | — | |
QYBQUVMLHHTKNO
|
6.6 | IC50 | 2 | — | |
RVHAEPLNTRENOO
|
6.6 | IC50 | 7 | — | |
RVJLYMOGPFRCQZ
|
6.6 | IC50 | 8 | — | |
SNEOQNDRTVGPGR
|
6.6 | IC50 | 7 | — | |
SXMMHTKZUYOEJX
|
6.6 | IC50 | 7 | — | |
XRNXDWRXNVCTGN
|
6.6 | IC50 | 7 | — | |
YECFQQVVMJBGDA
|
6.6 | IC50 | 7 | — | |
ZHOYYYIBRLNRRU
|
6.6 | IC50 | 7 | — | |
ZZVZQPYKDRXMAS
|
6.6 | IC50 | 7 | — | |
KHWWVAVHHRPPQY
|
6.6 | IC50 | 2 | — | |
SJNBIFGZSLRWRN
|
6.6 | IC50 | 2 | — | |
ACDXDMYMPLFVBN
|
6.6 | IC50 | 2 | — | |
OVPNQJVDAFNBDN
|
6.6 | Kd | 44 | Yes | |
ZULSMIQPZXUJHT
|
6.6 | IC50 | 2 | — | |
ZIBUGCUQIGHODU
|
6.6 | IC50 | 2 | — | |
UYYZTTPXKIYERF
|
6.6 | IC50 | 3 | — | |
VQPODCQNXLPCBS
|
6.6 | IC50 | 3 | — | |
VQUQBABVYFSBGV
|
6.5 | IC50 | 6 | — | |
JXVLTDGQDFESCZ
|
6.5 | IC50 | 7 | — | |
CEXGJBJPUFDWAH
|
6.5 | IC50 | 2 | — | |
CUNVHFMIKBBAIC
|
6.5 | Kd | 3 | — | |
DLISTLYUFVETPG
|
6.5 | IC50 | 7 | — | |
AJCFYLHZMCTQJH
|
6.5 | IC50 | 3 | — | |
YDLMQUFPYQIYTL
|
6.5 | IC50 | 2 | — | |
RHMNPYQXRSSRBE
|
6.5 | IC50 | 2 | — | |
UIJIOQITSXYSKV
|
6.5 | IC50 | 2 | — | |
MBFRPRCYZAVISU
|
6.4 | IC50 | 4 | — |