Target Details
| UniProt AC | Q9NYV4 |
|---|---|
| Gene Symbol | CDK12 |
| Protein Name | Cyclin-dependent kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 687
- Clinical molecules 4
- Avg pChEMBL 6.75
Active Molecules (687)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ITYQBQOTUYAYCQ
|
9.0 | IC50 | 2 | — | |
WMSVKCBXAUZFAL
|
9.0 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
9.0 | Kd | 599 | — | |
WPFIXUQBABAPHV
|
8.7 | IC50 | 2 | — | |
ADBAHGUKYCECGO
|
8.5 | IC50 | 2 | — | |
RAEQNTCTGLRWLL
|
8.5 | IC50 | 2 | — | |
UCBXGDNAAUVBDT
|
8.5 | IC50 | 2 | — | |
LYDGUMUGCXAMES
|
8.2 | IC50 | 2 | — | |
YJOJMGTVKMABKQ
|
8.2 | IC50 | 2 | — | |
GNLAZAPFJRZHHU
|
8.1 | IC50 | 2 | — | |
GVXKUINUYLVQFZ
|
8.1 | IC50 | 2 | — | |
CELWTMJZHQOTJD
|
8.0 | IC50 | 2 | — | |
KEWSSFSLZFTZRZ
|
8.0 | IC50 | 2 | — | |
YRNFLVUMZIRYKY
|
8.0 | IC50 | 2 | — | |
HIGWYWKMSCJGRM
|
8.0 | IC50 | 2 | — | |
FNRJTMUROZAOIB
|
7.9 | IC50 | 4 | — | |
FWCRSXACMNJQSL
|
7.9 | IC50 | 2 | — | |
HXKPNDMPSKRYFH
|
7.8 | IC50 | 3 | — | |
YEKKFBQFUXNWHX
|
7.8 | IC50 | 2 | — | |
NUMHIIKAGFNIFT
|
7.8 | IC50 | 8 | — | |
UVXKAHKGJDUTIP
|
7.8 | Kd | 3 | — | |
ZTNBFECBIFWCLE
|
7.8 | IC50 | 2 | — | |
ZYODEJHDTSBYGO
|
7.7 | IC50 | 2 | — | |
ALPNZWTZGINNPH
|
7.7 | IC50 | 6 | — | |
CEBRSPUCLVLGST
|
7.7 | IC50 | 6 | — | |
CHJCVDBWTBLBFK
|
7.7 | IC50 | 6 | — | |
COLFCNVHYZPNJS
|
7.7 | IC50 | 6 | — | |
CTTRZYCHOADLNP
|
7.7 | IC50 | 6 | — | |
CURXSSAFCGLCFN
|
7.7 | IC50 | 6 | — | |
IVVMEAPLRJRWHE
|
7.7 | IC50 | 9 | — | |
KSAUNOLTTIRZDD
|
7.7 | IC50 | 6 | — | |
LUWMNXZGQKQPGP
|
7.7 | IC50 | 6 | — | |
NCMNRWSGPFZNOJ
|
7.7 | IC50 | 6 | — | |
OASLPDKMYRJPOZ
|
7.7 | IC50 | 6 | — | |
QPXJKYBERAQULM
|
7.7 | IC50 | 6 | — | |
QWTLJZSIFBCFBX
|
7.7 | IC50 | 6 | — | |
RSEOXWPUDYEWFU
|
7.7 | IC50 | 6 | — | |
VAEFZVFYTXWCQB
|
7.7 | IC50 | 6 | — | |
VARHZJVBOVJDPK
|
7.7 | IC50 | 9 | — | |
WMWJOZFPAJCSFJ
|
7.7 | IC50 | 6 | — | |
XUBDCIJPSUUTBA
|
7.7 | IC50 | 6 | — | |
NBHWQTWPQQUECJ
|
7.7 | IC50 | 2 | — | |
REHJJRNUKGYLLU
|
7.7 | IC50 | 2 | — | |
RXPRVDHTUVMMTP
|
7.7 | IC50 | 2 | — | |
UWTHXCXQCZZLMX
|
7.7 | IC50 | 2 | — | |
GQAGWENJBMJZCO
|
7.6 | IC50 | 2 | — | |
KHKXXHNYGJSZMW
|
7.6 | IC50 | 2 | — | |
NHKBTLJNHPJRTH
|
7.6 | IC50 | 2 | — | |
XRMFYNTXRQPSMN
|
7.6 | IC50 | 2 | — | |
QVBVFLKFEISMLZ
|
7.6 | IC50 | 9 | — |