Target Details
| UniProt AC | Q9NYL2 |
|---|---|
| Gene Symbol | MAP3K20 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 20 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF07647 (SAM_2) |
Summary
- Multi-target molecules 117
- Clinical molecules 9
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (117)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QXRJBJVCBQSLTA
|
6.1 | Ki | 29 | — | |
RYYNGWLOYLRZLK
|
6.1 | Ki | 104 | — | |
UDFDIIVNIYWXDM
|
6.1 | Ki | 74 | — | |
XCHWBXBDZRJVDP
|
6.1 | Ki | 51 | — | |
ZLVOTRRGLSDLPF
|
6.1 | Ki | 36 | — | |
MVCOAUNKQVWQHZ
|
6.1 | Kd | 54 | Yes | |
WVUNYSQLFKLYNI
|
6.1 | Kd | 46 | Yes | |
HXNUFFCHRIWTRZ
|
6.0 | IC50 | 5 | — | |
DKNUPRMJNUQNHR
|
6.0 | Kd | 33 | — | |
IMHKMKWSWHFKTM
|
6.0 | Ki | 13 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MFMXAWQGPQXDRJ
|
6.0 | Ki | 27 | — | |
VLEFVPMCVJDTHZ
|
6.0 | Ki | 13 | — | |
ZGDSBEUMPIMXBM
|
6.0 | Ki | 42 | — | |
ZVWRFVCNQOECJS
|
6.0 | Ki | 71 | — |