Target Details
| UniProt AC | Q9NYL2 |
|---|---|
| Gene Symbol | MAP3K20 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 20 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF07647 (SAM_2) |
Summary
- Multi-target molecules 117
- Clinical molecules 9
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (117)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XFWUTMHVDGPWLH
|
6.8 | Ki | 75 | — | |
NNEJCBWOFHOVOJ
|
6.8 | IC50 | 2 | — | |
BFSMGDJOXZAERB
|
6.7 | Kd | 33 | — | |
WVXNSAVVKYZVOE
|
6.7 | IC50 | 92 | — | |
GCYXEGSPUDSZJY
|
6.7 | Ki | 82 | — | |
JSDGKSMNPHJDFK
|
6.7 | Ki | 35 | — | |
ULHGAQSVFPOUDY
|
6.7 | Ki | 43 | — | |
XKZQZMSAWVDRSP
|
6.7 | Ki | 39 | Yes | |
MIKAKZKNMYZLDX
|
6.6 | Ki | 42 | — | |
FNHKPVJBJVTLMP
|
6.6 | Kd | 29 | — | |
CSGQVNMSRKWUSH
|
6.5 | Kd | 21 | — | |
VAARYSWULJUGST
|
6.5 | Kd | 119 | Yes | |
KYACBMRLQMEIAI
|
6.5 | Ki | 30 | — | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
RKBYYWVZFBATHQ
|
6.5 | IC50 | 12 | — | |
UOOZSMNSBYVUGZ
|
6.4 | Ki | 32 | — | |
UUWNXFJBBYAMDT
|
6.4 | Ki | 46 | — | |
CUEAPAGGOWQGBA
|
6.4 | IC50 | 2 | — | |
LDOZZFMVGLMIQV
|
6.3 | IC50 | 2 | — | |
VWMJHAFYPMOMGF
|
6.3 | Kd | 15 | — | |
APPXQUDJLJXULP
|
6.3 | IC50 | 47 | — | |
UMBFDGUGXMOMHX
|
6.3 | IC50 | 12 | — | |
QFCXANHHBCGMAS
|
6.3 | Kd | 7 | — | |
KRIUNPBAQZGFQA
|
6.3 | Ki | 76 | — | |
OWDRQHVEJIYVOI
|
6.3 | Ki | 47 | — | |
OWRXHGAFWZFFCW
|
6.3 | Ki | 113 | — | |
RYAVJHIPOWNWDE
|
6.3 | Ki | 38 | — | |
WPHKIQPVPYJNAX
|
6.3 | Ki | 81 | — | |
JIOOBLLPEPCAAJ
|
6.3 | IC50 | 4 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
CKVWQORGCCEYHS
|
6.2 | Ki | 50 | — | |
NWAUBAGBGOPJLF
|
6.2 | Ki | 51 | Yes | |
OADRBDVURCEKRP
|
6.2 | Ki | 44 | — | |
XJSFDMGICAWQFS
|
6.2 | Ki | 60 | — | |
YEHCNYAQEBQCCS
|
6.2 | Ki | 74 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
ZCCPLJOKGAACRT
|
6.2 | Kd | 599 | — | |
SMPGEBOIKULBCT
|
6.2 | IC50 | 15 | — | |
UQRCJCNVNUFYDX
|
6.2 | Kd | 27 | — | |
SYCWRTUPLPDKDX
|
6.2 | IC50 | 3 | — | |
CMJCXYNUCSMDBY
|
6.1 | Kd | 15 | — | |
WJEOLQLKVOPQFV
|
6.1 | Kd | 24 | — | |
DKSNLQYRZJKYOC
|
6.1 | Ki | 51 | — | |
FGWOKLCRQJXPPQ
|
6.1 | Ki | 14 | — | |
GUMBHNMWKMFKRT
|
6.1 | Ki | 23 | — | |
HEKAIDKUDLCBRU
|
6.1 | Ki | 20 | — | |
KNACLJBHKVSTDL
|
6.1 | Ki | 40 | — | |
LXVBELDBJGYFEM
|
6.1 | Ki | 20 | — | |
MQRDVGBWWVWMEN
|
6.1 | Ki | 47 | — | |
PPCNMZPSQZFFGM
|
6.1 | Ki | 8 | — |