Target Details
| UniProt AC | Q9NYL2 |
|---|---|
| Gene Symbol | MAP3K20 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 20 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF07647 (SAM_2) |
Summary
- Multi-target molecules 117
- Clinical molecules 9
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (117)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DCJARECRZRVLPZ
|
8.7 | IC50 | 2 | — | |
XBRQXNKVCFFZSD
|
8.7 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
8.6 | Kd | 153 | — | |
UHROCBRCFGCHAX
|
8.6 | IC50 | 2 | — | |
BXSNWDRZYFXOFK
|
8.5 | IC50 | 2 | — | |
NZJCXRPMZJGVCC
|
8.5 | IC50 | 8 | — | |
SJSNJRWAMPFWPW
|
8.5 | IC50 | 2 | — | |
HLUOHTWAGISGKV
|
8.4 | IC50 | 2 | — | |
RCRNSDSDZVDENT
|
8.4 | IC50 | 2 | — | |
AWNCDMZXFFDAEU
|
8.4 | IC50 | 2 | — | |
QDSIBBLWWQMLJU
|
8.3 | IC50 | 2 | — | |
CRJDQLQMEZZQLC
|
8.2 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
8.2 | Kd | 85 | Yes | |
RDDZCQXKIJXMQN
|
8.2 | IC50 | 2 | — | |
NEDXWYOBFJNWEA
|
8.1 | IC50 | 2 | — | |
QRDCOOSKIFYKIQ
|
8.1 | Kd | 8 | — | |
RAHBGWKEPAQNFF
|
8.1 | Kd | 26 | — | |
UPJZIJDYXTYCDV
|
8.0 | Kd | 5 | — | |
PPILDDFMLSKYDE
|
8.0 | IC50 | 2 | — | |
HHZIURLSWUIHRB
|
8.0 | Kd | 57 | Yes | |
BTVPMDAMCUGYJV
|
7.9 | IC50 | 4 | — | |
NPVYSKNKKIWWJD
|
7.7 | IC50 | 2 | — | |
WPXVVAWAHQHJPF
|
7.7 | IC50 | 41 | — | |
GPXBXXGIAQBQNI
|
7.6 | IC50 | 11 | — | |
CXBBWVXSZINRCS
|
7.5 | Ki | 41 | — | |
HHCBMISMPSAZBF
|
7.4 | IC50 | 23 | — | |
PHXJVRSECIGDHY
|
7.4 | Kd | 59 | — | |
YZDJQTHVDDOVHR
|
7.4 | Kd | 23 | — | |
SEJGTFPOEJWEGG
|
7.3 | Kd | 149 | — | |
ZBNZXTGUTAYRHI
|
7.3 | Kd | 102 | Yes | |
KIGXQRBUVDDSPP
|
7.3 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
7.3 | Kd | 154 | — | |
JZXBVXNVBPKJRB
|
7.3 | IC50 | 2 | — | |
BGASXKCQPAUFOH
|
7.3 | IC50 | 2 | — | |
YABJJWZLRMPFSI
|
7.2 | Kd | 34 | — | |
ZGBAJMQHJDFTQJ
|
7.2 | Kd | 15 | — | |
PPCIDOUXWYIBPO
|
7.1 | IC50 | 6 | — | |
UBPYILGKFZZVDX
|
7.1 | Kd | 130 | Yes | |
XTUAHPVXWFQDFX
|
7.1 | IC50 | 2 | — | |
WKKRGQXAOQBWDF
|
7.0 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
7.0 | Kd | 112 | — | |
MCCCQFAOMZMZKE
|
7.0 | Ki | 52 | — | |
SRUYMJRFVGLQDV
|
7.0 | Ki | 37 | — | |
CYCZSOQHBKKPCR
|
7.0 | IC50 | 2 | — | |
PFTXFNSHFZLJNT
|
7.0 | IC50 | 17 | — | |
WJTJZDOMFKCYEA
|
6.9 | Kd | 6 | — | |
XLFJEGWLJGWRSM
|
6.9 | IC50 | 4 | — | |
NFMGZVPRGVERNN
|
6.8 | Ki | 44 | — | |
RJZDECGDCKOHBV
|
6.8 | Ki | 70 | — | |
WFTZMAAMCVPJJT
|
6.8 | Ki | 26 | — |