Target Details
| UniProt AC | Q9NY47 |
|---|---|
| Gene Symbol | CACNA2D2 |
| Protein Name | Voltage-dependent calcium channel subunit alpha-2/delta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08473 (VGCC_alpha2) PF00092 (VWA) PF08399 (VWA_N) |
Summary
- Multi-target molecules 63
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (63)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XCEJVZUIMKOKDS
|
6.7 | IC50 | 2 | — | |
GPVQFLNMUGKFCX
|
6.5 | IC50 | 2 | — | |
DXHGSDDDNQXAEJ
|
6.4 | IC50 | 26 | — | |
UXTXHFYVRKEMAW
|
6.4 | IC50 | 2 | — | |
XCLYWDHZGKKXTL
|
6.4 | IC50 | 2 | — | |
PSRVKIMUQGXDRE
|
6.3 | IC50 | 2 | — | |
CDPXETVZRHNLTM
|
6.2 | IC50 | 3 | — | |
INGBKPUFSDYYRV
|
6.2 | IC50 | 2 | — | |
JWUFFURPSKRHTA
|
6.1 | IC50 | 2 | — | |
PTYOAOCUXNHRIN
|
6.1 | IC50 | 2 | — | |
XKDFZZUFCHOVRN
|
6.1 | IC50 | 27 | — | |
GEHGVVUONLLQIR
|
6.0 | IC50 | 2 | — | |
JKAOGJXEFQNYHE
|
6.0 | IC50 | 2 | — |