Target Details
| UniProt AC | Q9NY46 |
|---|---|
| Gene Symbol | SCN3A |
| Protein Name | Sodium channel protein type 3 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 30
- Clinical molecules 4
- Avg pChEMBL 6.83
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CFMYXEVWODSLAX
|
8.3 | IC50 | 8 | — | |
ZUXRUQOEFBOTGF
|
8.0 | IC50 | 4 | — | |
FXTBLDWXLZMPPV
|
7.9 | IC50 | 3 | — | |
RPQXVSUAYFXFJA
|
7.9 | IC50 | 8 | — | |
LYTCVQQGCSNFJU
|
7.8 | IC50 | 3 | — | |
URSQNPPONHUJDL
|
7.8 | IC50 | 3 | — | |
TVQFYGIEBVVYRN
|
7.7 | IC50 | 4 | — | |
XOYPCMZEMYSCQC
|
7.7 | IC50 | 2 | — | |
XOAUGYVLRSCGBG
|
7.6 | IC50 | 8 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
KQQXPTRMUYKUIC
|
7.0 | Kd | 8 | — | |
KYBPOTYVFWNSGS
|
6.7 | Kd | 8 | — | |
DFBDAHMZXJYZJG
|
6.7 | IC50 | 7 | — | |
RDOIQAHITMMDAJ
|
6.6 | IC50 | 13 | — | |
WPYGCZCMGMVGNO
|
6.5 | IC50 | 4 | — | |
KUEGRSXKAHKHIA
|
6.5 | IC50 | 5 | — | |
IFFPICMESYHZPQ
|
6.5 | IC50 | 4 | — | |
QLKAFHZJICDACE
|
6.5 | IC50 | 3 | — | |
DERZBLKQOCDDDZ
|
6.4 | IC50 | 20 | Yes | |
KGGQAIGGEXFULW
|
6.3 | IC50 | 3 | — | |
DKGZKTPJOSAWFA
|
6.2 | IC50 | 21 | — | |
QVZCXCJXTMIDME
|
6.2 | IC50 | 4 | — | |
SMANXXCATUTDDT
|
6.2 | IC50 | 25 | Yes | |
CAFOIGUDKPQBIO
|
6.1 | IC50 | 3 | — | |
GKCBAIGFKIBETG
|
6.1 | IC50 | 10 | — | |
RMEDXOLNCUSCGS
|
6.1 | IC50 | 17 | Yes | |
PHSYVYPNRCSHQN
|
6.1 | IC50 | 3 | — | |
UIEATEWHFDRYRU
|
6.1 | IC50 | 8 | — | |
HBNPJJILLOYFJU
|
6.0 | IC50 | 21 | — | |
JJCFRYNCJDLXIK
|
6.0 | IC50 | 25 | Yes |