Target Details
| UniProt AC | Q9NXG6 |
|---|---|
| Gene Symbol | P4HTM |
| Protein Name | Transmembrane prolyl 4-hydroxylase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13640 (2OG-FeII_Oxy_3) PF13499 (EF-hand_7) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 7.87
Associated Diseases (1)
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDZRYLPROGBZMB
|
8.4 | IC50 | 8 | — | |
LYJKMVFAIXOQLE
|
8.3 | IC50 | 9 | — | |
NZTPJNIILSLMRH
|
8.2 | IC50 | 7 | — | |
QXQGSOMQKZFIRY
|
8.0 | IC50 | 10 | — | |
BJLOBSMGZUMYOP
|
7.8 | IC50 | 8 | — | |
NKWSAYGUIMPROA
|
7.6 | IC50 | 10 | — | |
KVQMUHHSWICEIH
|
6.7 | IC50 | 2 | — |