Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHPFQRTVUDXWCC
|
6.1 | Ki | 35 | — | |
KTEIFNKAUNYNJU
|
6.1 | Ki | 48 | — | |
QAJPIJHWTGPUNZ
|
6.1 | Ki | 37 | — | |
RWKDVIAVTRRJIR
|
6.1 | Ki | 23 | — | |
SPMHGQZFMNZCBV
|
6.1 | Ki | 30 | Yes | |
UOVCGJXDGOGOCZ
|
6.1 | Ki | 59 | — | |
VXYDJXMHISGSDA
|
6.1 | Ki | 59 | — | |
XSRHBCYNCKAFKS
|
6.1 | Ki | 45 | — | |
YWTBGJGMTBHQTM
|
6.1 | Ki | 65 | — | |
ZVWRFVCNQOECJS
|
6.1 | Ki | 71 | — | |
XZXHXSATPCNXJR
|
6.1 | Kd | 165 | Yes | |
ACJQMCQTSXRKNU
|
6.1 | IC50 | 2 | — | |
KICOSYRVTXVGTJ
|
6.1 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
IMRNKQWAMWWEKR
|
6.1 | IC50 | 5 | — | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
PBCZSGKMGDDXIJ
|
6.0 | Kd | 68 | Yes | |
OKKXBHWKOBOMGK
|
6.0 | Ki | 2 | — | |
AYJBHLUSGLQYDG
|
6.0 | Ki | 16 | — | |
BLUHZSPELLCJKH
|
6.0 | Ki | 9 | — | |
BPNUQXPIQBZCMR
|
6.0 | Ki | 60 | — | |
HDEZJSLYUKYKAZ
|
6.0 | Ki | 6 | — | |
HEUSUIRCBWROMH
|
6.0 | Ki | 64 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JVAFTPDILUBIGR
|
6.0 | IC50 | 9 | Yes | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NLUPJKQOKWBWFC
|
6.0 | Ki | 69 | — | |
WINHZLLDWRZWRT
|
6.0 | Ki | 66 | — | |
WUWDLXZGHZSWQZ
|
6.0 | Ki | 41 | — | |
YJBNTRQKJQHMTM
|
6.0 | Ki | 11 | — |