Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JXSBVAFKVRLTBE
|
6.3 | IC50 | 2 | — | |
JYXZRFURTZGRAR
|
6.3 | IC50 | 2 | — | |
JZUXTONNGLAGNS
|
6.3 | IC50 | 2 | — | |
KDEVAODGQITDKB
|
6.3 | IC50 | 2 | — | |
KJGJMKXKURZKFH
|
6.3 | IC50 | 2 | — | |
LKLKMYFYHDFSLS
|
6.3 | IC50 | 2 | — | |
OWGPCYDHMUISML
|
6.3 | IC50 | 2 | — | |
QJYCHNPBBAGVAL
|
6.3 | IC50 | 2 | — | |
RPMCQWGLLTVGAY
|
6.3 | IC50 | 2 | — | |
RWRVISCWYIIYAX
|
6.3 | IC50 | 2 | — | |
SDMRQHXJQFKDHV
|
6.3 | IC50 | 2 | — | |
UTBPPDSKJWJGTI
|
6.3 | IC50 | 2 | — | |
VLQGQOAWWLQXOZ
|
6.3 | IC50 | 2 | — | |
VZTDACMGWBXNRQ
|
6.3 | IC50 | 2 | — | |
WHFKPHNLHTXXRK
|
6.3 | IC50 | 2 | — | |
WJPDPEBXKRAWLO
|
6.3 | IC50 | 2 | — | |
WMPBJANDRBQKLJ
|
6.3 | IC50 | 2 | — | |
WUGZCFHBTBZAKK
|
6.3 | IC50 | 2 | — | |
WWNTVVYKRQBYEQ
|
6.3 | IC50 | 2 | — | |
XHWNTEWYWFMZBL
|
6.3 | IC50 | 2 | — | |
XMDZLJRPNPTNNM
|
6.3 | IC50 | 2 | — | |
XRKNHCDVUQOHPG
|
6.3 | IC50 | 2 | — | |
XSSXUEALEQDOGI
|
6.3 | IC50 | 2 | — | |
YLQBHUZSTBTNCJ
|
6.3 | IC50 | 2 | — | |
ZGPAYCQEDZYSFA
|
6.3 | IC50 | 2 | — | |
ZOPDRRJPLQTJDQ
|
6.3 | IC50 | 2 | — | |
ZRJZIWDFCSJDNF
|
6.3 | IC50 | 2 | — | |
ZVVNQPGCNBMROC
|
6.3 | IC50 | 2 | — | |
ZXICHULZXNAPKS
|
6.3 | IC50 | 2 | — | |
ZZPZTQIZEUBASL
|
6.3 | IC50 | 2 | — | |
DJVYXMINSBMUHH
|
6.2 | IC50 | 3 | — | |
LCHQFTFHRSXLRC
|
6.2 | IC50 | 2 | — | |
NHLRQGPSAURBBL
|
6.2 | IC50 | 3 | — | |
AGYZUONRISUOIK
|
6.2 | Ki | 10 | — | |
FDVSOQRNTAPCHB
|
6.2 | Ki | 40 | — | |
FMPKTXNCNJCHCC
|
6.2 | Ki | 25 | — | |
IOBVCHJTLVPPBR
|
6.2 | Ki | 39 | — | |
RKUKAACYUCUJEE
|
6.2 | Ki | 58 | — | |
VIZWJTHWUUQVGO
|
6.2 | Ki | 9 | — | |
VUHZDNOPEVGHEO
|
6.2 | Ki | 29 | — | |
WYCBJBMCGVVCMY
|
6.2 | Ki | 8 | — | |
ZWVZORIKUNOTCS
|
6.2 | Ki | 69 | — | |
JVAFTPDILUBIGR
|
6.2 | IC50 | 7 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
DYYISJDEAFXAFE
|
6.1 | IC50 | 2 | — | |
IAQIZJLJAOFQPG
|
6.1 | IC50 | 2 | — | |
XGALLCVXEZPNRQ
|
6.1 | Kd | 39 | Yes | |
YAPIPGOLZSTISM
|
6.1 | IC50 | 3 | — | |
CLRFYTGANQZOBS
|
6.1 | Ki | 41 | — | |
DKTMRIORKQEKMU
|
6.1 | Ki | 10 | — |