Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHRNVFQJUUXQIG
|
6.5 | IC50 | 2 | — | |
OUJZYQBEFNDJQN
|
6.5 | Ki | 71 | — | |
OXMXTNDWZBEXAL
|
6.5 | Kd | 2 | — | |
DASFSPDIWCMVRW
|
6.5 | IC50 | 21 | — | |
KGMSWMZCIQWBHX
|
6.5 | IC50 | 3 | — | |
MUYFQIQEBJQOGI
|
6.5 | IC50 | 2 | — | |
XDLZXQLBNFDCPI
|
6.5 | Ki | 4 | Yes | |
FTBMREIZHCLTPN
|
6.4 | IC50 | 3 | — | |
MSYMSSQHTUWZDQ
|
6.4 | IC50 | 2 | — | |
WTUNZCQRKFMUHJ
|
6.4 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.4 | Kd | 599 | — | |
WAOZMJFYNREQLU
|
6.4 | IC50 | 2 | — | |
QTTGVGLTCILDCA
|
6.4 | IC50 | 7 | — | |
MLCCBIGYVHDJCI
|
6.4 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
6.4 | Ki | 54 | — | |
FONINLXADYUZFI
|
6.4 | Ki | 25 | — | |
HYNNWLVWJXWXFO
|
6.4 | IC50 | 2 | — | |
IMLXFZLHOPEBPM
|
6.4 | Ki | 12 | — | |
KCECLCOMITXYJK
|
6.4 | IC50 | 2 | — | |
LRINYHMQZRENCY
|
6.4 | Ki | 29 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
LYUCMSBGXASQAS
|
6.4 | IC50 | 2 | — | |
MZDKLVOWGIOKTN
|
6.4 | Ki | 80 | — | |
NKGLJTITEFZKAN
|
6.4 | Ki | 35 | — | |
OADRBDVURCEKRP
|
6.4 | Ki | 44 | — | |
QRCXMLQLNQMAFC
|
6.4 | Ki | 10 | — | |
UMTWTCVTRDYHQQ
|
6.4 | Ki | 56 | — | |
FELCCLMGXTVEGI
|
6.4 | Ki | 4 | Yes | |
ADLJEZREHNJMCU
|
6.4 | IC50 | 6 | — | |
GXJJTQDCWLONOL
|
6.4 | Ki | 6 | Yes | |
MHRNVFQJUUXQIG
|
6.3 | IC50 | 2 | — | |
CYJPFBCHYRZAJL
|
6.3 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
6.3 | IC50 | 130 | Yes | |
ZFIKQWONLNAODK
|
6.3 | IC50 | 2 | — | |
HWYGUNZPOCDUSM
|
6.3 | IC50 | 2 | — | |
IDGNCVHQDDOPND
|
6.3 | IC50 | 6 | — | |
PPIGWXNYCGUCMZ
|
6.3 | IC50 | 2 | — | |
CWBWMDSAVFJNAD
|
6.3 | Ki | 7 | — | |
RJZDECGDCKOHBV
|
6.3 | Ki | 70 | — | |
SUULIUKTZNKMMB
|
6.3 | Ki | 10 | — | |
UFMAIBLTWQRHAK
|
6.3 | Ki | 10 | — | |
AIYIKSZSMWXXLB
|
6.3 | IC50 | 2 | — | |
BTHHTUIURXXDQK
|
6.3 | IC50 | 2 | — | |
DIVBAVIPIJCFQU
|
6.3 | IC50 | 2 | — | |
FASAXWZUGXWYCH
|
6.3 | IC50 | 2 | — | |
FYPLNZXUWFDWFV
|
6.3 | IC50 | 2 | — | |
GKSLYGBWVIREPH
|
6.3 | IC50 | 2 | — | |
HCVYZVCMHVIECU
|
6.3 | IC50 | 2 | — | |
IOAFUECVQSRNGN
|
6.3 | IC50 | 2 | — | |
IQMFQXFGETWXJL
|
6.3 | IC50 | 2 | — |