Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJWADKUXOQKYQJ
|
6.9 | IC50 | 2 | — | |
CRSHGUZUNKJVIT
|
6.8 | IC50 | 2 | — | |
LRINILBKXCVIMV
|
6.8 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
MUYFQIQEBJQOGI
|
6.8 | IC50 | 2 | — | |
RGJUJSDOHVLJHD
|
6.8 | IC50 | 2 | — | |
VBIYDORVDCFKHM
|
6.8 | IC50 | 13 | — | |
CLEGDJQQHUTCOW
|
6.8 | Ki | 43 | — | |
GIRPCUVQSUVBEK
|
6.8 | IC50 | 3 | — | |
KRIUNPBAQZGFQA
|
6.8 | Ki | 76 | — | |
NJPWCTYVEJIQBM
|
6.8 | Ki | 72 | — | |
NXNQLECPAXXYTR
|
6.8 | Ki | 29 | — | |
PSCJSWRVCKUMSL
|
6.8 | Ki | 35 | — | |
RYYNGWLOYLRZLK
|
6.8 | Ki | 104 | — | |
SELXDFVNFMEQCP
|
6.8 | Ki | 5 | — | |
UZYWWOWQGPMEIC
|
6.8 | IC50 | 2 | — | |
FTFDOZLQPLTYBX
|
6.8 | IC50 | 7 | Yes | |
GHAHLIVGSBTTLD
|
6.8 | IC50 | 2 | — | |
HZYIMGKDYXEJDM
|
6.8 | IC50 | 3 | — | |
JBGWDRMZKMTPOT
|
6.8 | IC50 | 3 | — | |
SNKIPAIHEQSWBK
|
6.8 | IC50 | 2 | — | |
KKHYJYDEGGYOIC
|
6.7 | IC50 | 2 | — | |
DZIXRHJRLCGYPK
|
6.7 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
LKXQEHYYVXRDJC
|
6.7 | IC50 | 2 | — | |
GCBJDOWIQHMCMR
|
6.7 | Ki | 84 | — | |
KIUHBHFVVQQALF
|
6.7 | Ki | 9 | — | |
LOMGAGWJYPGDLT
|
6.7 | Ki | 8 | — | |
NRSGWEVTVGZDFC
|
6.7 | Ki | 50 | — | |
OLVBAUVSICCWEJ
|
6.7 | Ki | 39 | — | |
QTCFYQHZJIIHBS
|
6.7 | IC50 | 2 | — | |
UYJNQQDJUOUFQJ
|
6.7 | Ki | 68 | — | |
XOJQJDHWKVZUAT
|
6.7 | Ki | 9 | — | |
YUOWJICKAJQZLS
|
6.7 | Ki | 35 | — | |
ASEWBZJHLDHXLR
|
6.7 | Ki | 2 | — | |
QNABDSWBQJKBHK
|
6.7 | IC50 | 45 | — | |
XSIMOSPDULMWPL
|
6.7 | IC50 | 3 | — | |
YLJPQGVBJWZONC
|
6.6 | IC50 | 6 | — | |
BSFNGHCTZDCQBF
|
6.6 | Ki | 93 | — | |
FAYAUAZLLLJJGH
|
6.6 | Ki | 36 | Yes | |
NRZYTPAJGVTKIM
|
6.6 | Ki | 38 | — | |
OQHALFBQFMAXFZ
|
6.6 | Ki | 9 | — | |
SYLTYCLPHHSEIJ
|
6.6 | Ki | 27 | — | |
YMIJUBCSOKSFRU
|
6.6 | Ki | 87 | — | |
PWCLOPMRUGHLET
|
6.6 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
6.5 | Kd | 50 | — | |
TWWKXZDIDHDHRF
|
6.5 | IC50 | 7 | — | |
AUDNGNGLLRZLDR
|
6.5 | Ki | 33 | — | |
KEBXAEFZLCNLJJ
|
6.5 | Ki | 13 | — | |
KOHNRDPXFDZZJF
|
6.5 | Ki | 31 | — |