Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BRNMCVNQMQLRHM
|
7.3 | IC50 | 3 | — | |
GAIBRRPRULCSHG
|
7.3 | IC50 | 2 | — | |
LBBNQAJEJZYWPT
|
7.3 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
7.3 | Ki | 72 | — | |
AHYTYKPDDJPJKK
|
7.3 | IC50 | 2 | — | |
JMHQUQCLIVNTHT
|
7.3 | Ki | 24 | — | |
JZTOUVBEZONDKA
|
7.3 | Ki | 80 | — | |
YEHCNYAQEBQCCS
|
7.3 | Ki | 74 | — | |
LLYRJVQDZYKVCX
|
7.3 | IC50 | 2 | — | |
ZXPBSKBKOLENLI
|
7.3 | IC50 | 2 | — | |
SKDSRJRRAQLUPP
|
7.2 | IC50 | 8 | Yes | |
VCCDOPPWOSIMCD
|
7.2 | IC50 | 2 | — | |
AEWUMWRWGREICZ
|
7.2 | IC50 | 2 | — | |
RVSSNRBUPQUIEG
|
7.2 | IC50 | 5 | — | |
DYNHJHQFHQTFTP
|
7.2 | Kd | 38 | — | |
NBLFGELIWIKRAC
|
7.2 | Ki | 8 | — | |
NXCSPXHUVYRKQK
|
7.2 | IC50 | 2 | — | |
DSSNAGYVGTYAGH
|
7.2 | IC50 | 10 | — | |
UEFCSGDOOJJXTN
|
7.2 | IC50 | 46 | — | |
WINHZLLDWRZWRT
|
7.2 | Kd | 201 | Yes | |
PHXJVRSECIGDHY
|
7.2 | IC50 | 59 | — | |
ZCEVGIAITKATNG
|
7.2 | IC50 | 2 | — | |
JFKRMJRQGVELFG
|
7.1 | IC50 | 3 | — | |
FKNJKNHEBUMLTR
|
7.1 | IC50 | 2 | — | |
LJCSOVSRKPFJJG
|
7.1 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.1 | Kd | 170 | — | |
UHTHHESEBZOYNR
|
7.1 | Kd | 66 | Yes | |
YCFRZMCRPHNZOC
|
7.1 | IC50 | 7 | — | |
YCFRZMCRPHNZOC
|
7.1 | IC50 | 6 | — | |
QQWUGDVOUVUTOY
|
7.1 | Kd | 231 | Yes | |
XCHZMPYWMULFBJ
|
7.1 | Ki | 4 | Yes | |
JMQCXZBXWOIDIO
|
7.1 | Ki | 9 | — | |
BKDJJDIXKRUBLT
|
7.1 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
7.1 | Kd | 151 | — | |
UAIANIHUMMKHJR
|
7.1 | IC50 | 3 | — | |
SWPXADMCNLNAGW
|
7.0 | IC50 | 10 | — | |
OUCUNVKXSOPBBS
|
7.0 | IC50 | 4 | — | |
QYGMZFLXMWJYRJ
|
7.0 | Ki | 14 | — | |
RAIGSWRYTFZVQJ
|
7.0 | IC50 | 2 | — | |
XFWUTMHVDGPWLH
|
7.0 | Ki | 75 | — | |
TUAJTUKIIJXVON
|
7.0 | IC50 | 3 | — | |
VYOVIFUEUXGCRT
|
7.0 | IC50 | 2 | — | |
UIEHXCCYHAUOFD
|
7.0 | IC50 | 3 | — | |
NQZRHTLUKLOASK
|
6.9 | IC50 | 3 | — | |
FQVCSBNTPQDQSS
|
6.9 | IC50 | 3 | — | |
XPMRQKGHVCXNDM
|
6.9 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
6.9 | Ki | 70 | — | |
MVJMMLFMPWITEJ
|
6.9 | Ki | 110 | — | |
PIQCTGMSNWUMAF
|
6.9 | Kd | 137 | Yes | |
RVFYCRCCTDEQQD
|
6.9 | IC50 | 4 | — |