Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UDRXOUVRNMKWQA
|
7.8 | Ki | 8 | — | |
VDJSCKUWUKCUEK
|
7.8 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
7.8 | IC50 | 46 | — | |
QRRAWPZSLULASL
|
7.8 | IC50 | 2 | — | |
MIWFIZLZRBKGQU
|
7.7 | IC50 | 2 | — | |
SZURKEABSBIIMJ
|
7.7 | IC50 | 5 | — | |
VJDQIINVHIBHNW
|
7.7 | IC50 | 2 | — | |
VVQWKIHKNXGJKG
|
7.7 | IC50 | 2 | — | |
WANRGEOLLIFNBS
|
7.7 | IC50 | 4 | — | |
JJSAYYGWZQRZJC
|
7.7 | IC50 | 2 | — | |
SOQDSWCPJNRWBD
|
7.7 | IC50 | 2 | — | |
ILMYAITZJAJSEG
|
7.7 | IC50 | 2 | — | |
RAFFLDOJXQAJPF
|
7.7 | IC50 | 2 | — | |
NYYOAOHKRVOFGH
|
7.7 | IC50 | 5 | — | |
JANBIXNDYNRYQP
|
7.7 | IC50 | 2 | — | |
MJGKLMMMXSNBCX
|
7.7 | IC50 | 3 | — | |
QKXDICQFNATVHN
|
7.7 | IC50 | 3 | — | |
LYADGAGFYYXXIO
|
7.6 | IC50 | 82 | — | |
NXSJMRCTGYTSTK
|
7.6 | Kd | 200 | — | |
WRDPDAIOMMMLNR
|
7.6 | IC50 | 2 | — | |
HRNAVIYNHGZRMP
|
7.6 | IC50 | 3 | — | |
MURKOANUFGPGGP
|
7.6 | IC50 | 2 | — | |
OWIYRPIJTDKPDU
|
7.6 | IC50 | 2 | — | |
WGMWEVJCHUDPID
|
7.6 | IC50 | 2 | — | |
WZBIRANKKAOEQU
|
7.6 | IC50 | 2 | — | |
ZJOCDAGVCZOCSS
|
7.6 | IC50 | 2 | — | |
NANIKNNTSLTWED
|
7.6 | IC50 | 2 | — | |
PONZXJHPMSOTCH
|
7.6 | IC50 | 2 | — | |
BBKKFCZZAZLULJ
|
7.6 | IC50 | 2 | — | |
FQBRQRVXPUQKLG
|
7.5 | IC50 | 10 | — | |
AYLVCUFENDVPDV
|
7.5 | IC50 | 2 | — | |
BPTXXXCWMKGAFJ
|
7.5 | IC50 | 2 | — | |
OFYBGNCNPOQMEB
|
7.5 | IC50 | 2 | — | |
RBTVHFPPQWRMEB
|
7.5 | IC50 | 2 | — | |
ITDPQZHRPNERLI
|
7.5 | IC50 | 3 | — | |
FLEAYYMORDPWAJ
|
7.5 | Ki | 90 | — | |
CDAIGUSYJLTHBH
|
7.5 | IC50 | 2 | — | |
JYDDZHVWLDZGJX
|
7.5 | IC50 | 2 | — | |
QYZYODZZZGIMSS
|
7.4 | Ki | 2 | — | |
KEAPLOABAMRRFQ
|
7.4 | IC50 | 2 | — | |
AZIKDQBYCZVPSU
|
7.4 | IC50 | 3 | — | |
YBPNMUVFLXIRNQ
|
7.4 | IC50 | 2 | — | |
IBJBVUBNAOGQIK
|
7.4 | IC50 | 2 | — | |
FUMCKNCUEAQHCV
|
7.4 | Ki | 103 | — | |
OFPXYNMQWVCVKZ
|
7.4 | Ki | 8 | — | |
OXRQZPOYHSRCIB
|
7.4 | IC50 | 3 | — | |
SNCZIVUNTWOQAF
|
7.4 | IC50 | 4 | — | |
VSNJCPXJAHKLRS
|
7.4 | Ki | 7 | Yes | |
DTHDBWPUQXSBEE
|
7.4 | IC50 | 3 | — | |
FQGLEOSEPJEJPE
|
7.4 | IC50 | 2 | — |