Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DWDATRBHPMAHRD
|
8.2 | IC50 | 2 | — | |
CGZANCKEFIHBJE
|
8.2 | IC50 | 2 | — | |
HXUCFPZSRWJRRN
|
8.2 | IC50 | 3 | — | |
RDTAHMIMQLRAMR
|
8.2 | IC50 | 2 | — | |
UUSDUSGMWIXJOT
|
8.2 | IC50 | 2 | — | |
YEZSPJXJBLNYQO
|
8.2 | IC50 | 3 | — | |
MURKOANUFGPGGP
|
8.2 | IC50 | 2 | — | |
PSBLEKZDHVNIQM
|
8.1 | IC50 | 2 | — | |
VZOLINZYKOLXAC
|
8.1 | IC50 | 2 | — | |
VZOLINZYKOLXAC
|
8.1 | IC50 | 2 | — | |
FEJCKYYKSNIWCL
|
8.1 | IC50 | 2 | — | |
BUJSZRICYLPWCM
|
8.1 | IC50 | 3 | — | |
BUZQLQAPFVMMQY
|
8.1 | IC50 | 2 | — | |
RHGZQGXELRMGES
|
8.1 | IC50 | 8 | Yes | |
SKWDOWYVGZFBQX
|
8.1 | IC50 | 2 | — | |
AWEZXOKZISCYJP
|
8.1 | IC50 | 2 | — | |
IEOZVBDPTHRYGK
|
8.1 | Ki | 3 | — | |
PFCFMZHQWUDEEB
|
8.1 | IC50 | 2 | — | |
XAIKPAUBEILQRY
|
8.1 | IC50 | 2 | — | |
HHVUHFYJIYORJI
|
8.1 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
8.1 | Kd | 88 | Yes | |
RRQPKDCUEZDZOV
|
8.1 | IC50 | 2 | — | |
SZFYZDIPRMLBDC
|
8.1 | IC50 | 9 | — | |
UJFKYOVASOKVMM
|
8.1 | IC50 | 2 | — | |
UZYWWOWQGPMEIC
|
8.1 | IC50 | 2 | — | |
WHCMKDGCCYRJKV
|
8.1 | IC50 | 2 | — | |
YUANXHKOYHEHOW
|
8.1 | IC50 | 2 | — | |
APNCLDVFDSDLCS
|
8.0 | IC50 | 2 | — | |
DURNYYKOVXELMP
|
8.0 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.0 | Ki | 118 | — | |
ONRYANARCHPXRQ
|
8.0 | IC50 | 2 | — | |
SMIIJPDEPOIIHO
|
8.0 | IC50 | 2 | — | |
ZDIREJTXQKRZCD
|
8.0 | IC50 | 2 | — | |
MURKOANUFGPGGP
|
8.0 | IC50 | 2 | — | |
WGQUSQTWZRXHGK
|
8.0 | IC50 | 3 | — | |
HRNKXLATVXBONQ
|
7.9 | IC50 | 2 | — | |
IYZWULIJOWJSKT
|
7.9 | IC50 | 2 | — | |
NTKWIHLGLPIAOG
|
7.9 | IC50 | 2 | — | |
OWSBCGNMLGHERL
|
7.9 | IC50 | 2 | — | |
SFXNZFNSPSLHEA
|
7.9 | IC50 | 2 | — | |
JAMDNXUAYUHJLJ
|
7.9 | Ki | 40 | — | |
VWVYILCFSYNJHF
|
7.9 | Ki | 49 | — | |
ZFLJQOGIHBIDNZ
|
7.9 | IC50 | 2 | — | |
RPGMSHCJIWHISY
|
7.9 | IC50 | 3 | — | |
RPGMSHCJIWHISY
|
7.9 | IC50 | 3 | — | |
OACJMCGKLHFOLN
|
7.8 | IC50 | 2 | — | |
VMYCKCWYEIGQOV
|
7.8 | IC50 | 3 | — | |
MXCUSZDSXDTMHC
|
7.8 | IC50 | 3 | — | |
XPMRQKGHVCXNDM
|
7.8 | IC50 | 2 | — | |
GDYZFFBMSBDTAA
|
7.8 | Ki | 60 | — |