Target Details
| UniProt AC | Q9NWZ3 |
|---|---|
| Gene Symbol | IRAK4 |
| Protein Name | Interleukin-1 receptor-associated kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 431
- Clinical molecules 21
- Avg pChEMBL 7.37
KEGG Pathways (22)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Influenza A
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Associated Diseases (1)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TZUYQGIZCUHALE
|
9.0 | IC50 | 2 | — | |
UZBFFCBUJQNOPY
|
9.0 | IC50 | 3 | — | |
XBMMPGPTZWUPAP
|
9.0 | IC50 | 2 | — | |
XMWONVHOMANOOY
|
9.0 | IC50 | 3 | — | |
CEAYRKIZESVQSN
|
8.9 | Ki | 4 | — | |
DQEKCEBMQCYICP
|
8.9 | Ki | 3 | — | |
ATVTUVKVZSYFBE
|
8.8 | IC50 | 7 | — | |
UIARLYUEJFELEN
|
8.8 | Kd | 289 | Yes | |
BFBOXYLGKAPSFY
|
8.7 | IC50 | 2 | — | |
CMKUJKFQBWYWBJ
|
8.7 | IC50 | 3 | — | |
FUOKGTYXSNVQIW
|
8.7 | IC50 | 3 | — | |
HXYSWTZEQZNVDR
|
8.7 | IC50 | 3 | — | |
KSJNXKBKMYLRSO
|
8.7 | IC50 | 3 | — | |
LVDGPLKQEUXHAV
|
8.7 | IC50 | 2 | — | |
MEBULVBTXSYJKD
|
8.7 | IC50 | 3 | — | |
OSATXCGVOWUMIG
|
8.7 | IC50 | 2 | — | |
PKAXKMPZRBQIOO
|
8.7 | IC50 | 3 | — | |
RDBXDKAXTSZQAP
|
8.7 | IC50 | 2 | — | |
SLKSOMMHRLEOCJ
|
8.7 | IC50 | 2 | — | |
VBVMZSHPPUKQDJ
|
8.7 | IC50 | 2 | — | |
YMEYAMDEQBMREG
|
8.7 | IC50 | 3 | — | |
CVWXJKQAOSCOAB
|
8.7 | IC50 | 35 | — | |
RKDBBXGRXIYXMB
|
8.7 | Kd | 2 | — | |
CLRGCYMGDBZQTB
|
8.6 | Ki | 2 | — | |
DGUFRRJUHIZTQE
|
8.6 | Ki | 3 | — | |
FLZAOAIEJUXTAH
|
8.5 | IC50 | 2 | — | |
IWIYCPMVAVQALP
|
8.5 | IC50 | 2 | — | |
KLAHVJUJQYVKPO
|
8.5 | IC50 | 2 | — | |
OCDYJTRAVKONSS
|
8.5 | IC50 | 3 | — | |
OTAZAWFIQUEVLG
|
8.5 | IC50 | 3 | — | |
PQMBTEFIJYDBHA
|
8.5 | IC50 | 2 | — | |
UBKAKYFRDGQVJG
|
8.5 | IC50 | 3 | — | |
YTQVSNUZNYHPOL
|
8.5 | Kd | 2 | — | |
QQIQOMIKWUAMAA
|
8.4 | IC50 | 7 | — | |
CEOQQVRJCFJERM
|
8.4 | IC50 | 2 | — | |
DPRNXTSMYVCYLJ
|
8.4 | IC50 | 13 | — | |
DUOPMZXNVCHSKJ
|
8.4 | IC50 | 3 | — | |
OWRXHGAFWZFFCW
|
8.4 | Ki | 113 | — | |
QJGDGWJGAAATCO
|
8.4 | IC50 | 2 | — | |
YZPJEKZOTFSOHR
|
8.4 | IC50 | 2 | — | |
DVRHHNDPHSXUFJ
|
8.4 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.3 | IC50 | 408 | — | |
DJVYXMINSBMUHH
|
8.3 | IC50 | 8 | — | |
DJVYXMINSBMUHH
|
8.3 | IC50 | 8 | — | |
HXEIWJBTKNXMHO
|
8.3 | IC50 | 2 | — | |
IBYHNCOWDYTTRQ
|
8.3 | IC50 | 2 | — | |
KYNJAMYDYPTYDZ
|
8.3 | IC50 | 2 | — | |
XPHWIERLJBFPFV
|
8.3 | Ki | 69 | — | |
ZOGZUMFMIBABFJ
|
8.3 | IC50 | 2 | — | |
FXKMVTAKVQDJJT
|
8.3 | IC50 | 2 | — |