Target Details
| UniProt AC | Q9NUW8 |
|---|---|
| Gene Symbol | TDP1 |
| Protein Name | Tyrosyl-DNA phosphodiesterase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF06087 (Tyr-DNA_phospho) |
Summary
- Multi-target molecules 4
- Clinical molecules 0
- Avg pChEMBL 6.89
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GIXWDMTZECRIJT
|
7.8 | IC50 | 9 | — | |
VWTPGUPXPKYBNL
|
7.8 | IC50 | 8 | — | |
RJTFJQBDICKHOW
|
6.0 | IC50 | 2 | — | |
ZJHZBDRZEZEDGB
|
6.0 | IC50 | 3 | — |