Target Details
| UniProt AC | Q9NSY1 |
|---|---|
| Gene Symbol | BMP2K |
| Protein Name | BMP-2-inducible protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15282 (BMP2K_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 111
- Clinical molecules 18
- Avg pChEMBL 7.15
KEGG Pathways (1)
Active Molecules (111)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MXOVNNMQDFPQKY
|
7.3 | Ki | 3 | — | |
PIQCTGMSNWUMAF
|
7.3 | Kd | 137 | Yes | |
IIKPYJZUOZRTIB
|
7.2 | Ki | 4 | — | |
GCIKSSRWRFVXBI
|
7.2 | Kd | 109 | Yes | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
INTMVZKGQXMUML
|
7.1 | Ki | 3 | — | |
HINOQCZIDBNXEI
|
7.0 | IC50 | 5 | — | |
KOZFSFOOLUUIGY
|
7.0 | Kd | 88 | Yes | |
CWDJCUXKEDKAQE
|
7.0 | IC50 | 2 | — | |
GGYXFRIDIFIYBO
|
7.0 | IC50 | 2 | — | |
HXRGDEBGHHKEEK
|
7.0 | IC50 | 2 | — | |
JAWYVNPEVKLENS
|
7.0 | IC50 | 2 | — | |
JKCNRFQYOHWEDM
|
7.0 | IC50 | 2 | — | |
MHWJYODTCNDXJW
|
7.0 | IC50 | 2 | — | |
NSQIWTMRSLRZLP
|
7.0 | IC50 | 2 | — | |
NTXHJAVJAVSTET
|
7.0 | IC50 | 2 | — | |
WSEPAQYPZMEAQP
|
7.0 | IC50 | 2 | — | |
YLVDJOXELSCRPM
|
7.0 | IC50 | 3 | — | |
BPNUQXPIQBZCMR
|
6.9 | Kd | 83 | Yes | |
GCTFTMWXZFLTRR
|
6.9 | IC50 | 7 | — | |
KMVVQXBUHOYQKZ
|
6.9 | Ki | 3 | — | |
GUBJNPWVIUFSTR
|
6.8 | Kd | 103 | — | |
FMNWOBLAZAYOSG
|
6.8 | IC50 | 5 | — | |
QTBWCSQGBMPECM
|
6.8 | Kd | 21 | Yes | |
HVHRHDHQHUAOQI
|
6.8 | IC50 | 5 | — | |
JTVBXQAYBIJXRP
|
6.8 | Kd | 20 | — | |
RKBMAROJKLHAMI
|
6.8 | IC50 | 6 | — | |
IAYGCINLNONXHY
|
6.7 | Kd | 50 | — | |
KDKUVYLMPJIGKA
|
6.7 | Kd | 91 | Yes | |
HFNKQEVNSGCOJV
|
6.7 | Kd | 65 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 91 | Yes | |
DKZYXHCYPUVGAF
|
6.6 | Kd | 112 | — | |
QHPJIUARPKBLQQ
|
6.6 | IC50 | 3 | — | |
NGBWQVJCOYTGOR
|
6.5 | IC50 | 8 | — | |
NHFDRBXTEDBWCZ
|
6.5 | Kd | 12 | Yes | |
JKCNRFQYOHWEDM
|
6.5 | IC50 | 2 | — | |
NSQIWTMRSLRZLP
|
6.5 | IC50 | 2 | — | |
RETYBSQLAYVBLT
|
6.5 | IC50 | 2 | — | |
STOKTXVQCBDPNW
|
6.5 | IC50 | 2 | — | |
WSEPAQYPZMEAQP
|
6.5 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
6.5 | Kd | 130 | Yes | |
QDITZBLZQQZVEE
|
6.4 | Kd | 19 | — | |
ZCBUQCWBWNUWSU
|
6.4 | Kd | 59 | — | |
ZHJGWYRLJUCMRT
|
6.3 | Kd | 18 | — | |
WVUNYSQLFKLYNI
|
6.3 | Kd | 46 | Yes | |
UJIAQDJKSXQLIT
|
6.2 | Kd | 38 | — | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
KTEIFNKAUNYNJU
|
6.1 | Kd | 114 | — | |
PBCZSGKMGDDXIJ
|
6.1 | Kd | 68 | Yes |